Compile Data Set for Download or QSAR
Report error Found 2928 for UniProtKB: O35433
LigandPNGBDBM20319(3-[(4-tert-butylphenyl)methyl]-1-[2-(4-methanesulf...)
Affinity DataEC50:  1.80E+3nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2008
Entry Details Article
PubMed
LigandPNGBDBM20334(1-isoquinolin-5-yl-3-{[4-(trifluoromethyl)phenyl]m...)
Affinity DataEC50:  24nMpH: 7.4 T: 2°CAssay Description:The functional antagonist activity of compounds at the TRPV1 receptor was determined with a Ca2+ influx assay by measuring the effect on capsaicin (0...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2008
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223199(CHEMBL290274)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223202(CHEMBL36669)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223203(CHEMBL39466)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223204(CHEMBL287757)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223205(CHEMBL39079)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223206(CHEMBL289694)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223207(CHEMBL39219)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM20284(N-[2-(4-chlorophenyl)ethyl]-7,8-dihydroxy-2,3,4,5-...)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223197(CHEMBL289068)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223200(CHEMBL291285)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223209(CHEMBL417334)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223201(CHEMBL440471)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223208(CHEMBL39199)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223213(CHEMBL38831)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223210(CHEMBL39785)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223198(CHEMBL39913)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223211(CHEMBL39289)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223212(CHEMBL39108)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223214(CHEMBL39817)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50223215(CHEMBL289693)
Affinity DataEC50: >1.00E+5nMAssay Description:Ability to cause [Ca2+] influx in neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
LigandPNGBDBM50196348(2-(3-(4-hydroxy-3-methoxybenzyl)thioureido)-4-(4-t...)
Affinity DataEC50:  22nMAssay Description:Agonist activity at rat TRPV1 expressed in CHO cells assessed as maximal calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50196337(2-((3-(4-hydroxy-3-methoxybenzyl)thioureido)methyl...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at rat TRPV1 expressed in CHO cells assessed as maximal calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50196334(2-(3-(4-hydroxy-3-methoxybenzyl)thioureido)-4-(3,4...)
Affinity DataEC50:  15nMAssay Description:Agonist activity at rat TRPV1 expressed in CHO cells assessed as maximal calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50440399(CHEMBL2425544)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at rat TRPV1 expressed in CHO cells assessed as stimulation of Ca2+ uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
LigandPNGBDBM50440402(CHEMBL2425547)
Affinity DataEC50:  5nMAssay Description:Agonist activity at rat TRPV1 expressed in CHO cells assessed as stimulation of Ca2+ uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
LigandPNGBDBM50440400(CHEMBL2425551)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity at rat TRPV1 expressed in CHO cells assessed as stimulation of Ca2+ uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
LigandPNGBDBM50440401(CHEMBL2425550)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at rat TRPV1 expressed in CHO cells assessed as stimulation of Ca2+ uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
LigandPNGBDBM50163238(4-Pyridin-4-yl-piperazine-1-carboxylic acid (4-chl...)
Affinity DataEC50:  3.60E+3nMAssay Description:Effective concentration against rat transient receptor potential vanilloid 1 receptor (n=6)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50163240(4-(2-Trifluoromethyl-phenyl)-piperazine-1-carboxyl...)
Affinity DataEC50:  1.28E+3nMAssay Description:Effective concentration against rat transient receptor potential vanilloid 1 receptor (n=3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50163232(4-(2-Trifluoromethyl-phenyl)-piperazine-1-carboxyl...)
Affinity DataEC50:  7.29E+3nMAssay Description:Effective concentration against rat transient receptor potential vanilloid 1 receptor (n=3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50163231(4-Pyridin-3-yl-piperazine-1-carboxylic acid (4-tri...)
Affinity DataEC50:  2.67E+3nMAssay Description:Effective concentration against rat transient receptor potential vanilloid 1 receptor (n=3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50163229(4-(2-Trifluoromethyl-phenyl)-piperazine-1-carboxyl...)
Affinity DataEC50:  275nMAssay Description:Effective concentration against rat transient receptor potential vanilloid 1 receptor (n=4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50163243(4-(2-Trifluoromethyl-phenyl)-piperazine-1-carboxyl...)
Affinity DataEC50:  8.30E+3nMAssay Description:Effective concentration against rat transient receptor potential vanilloid 1 receptor (n=6)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50163220(3-Methyl-3'',4'',5'',6''-tetrahydro-2''H-[2,4'']bi...)
Affinity DataEC50:  1.96E+3nMAssay Description:Effective concentration against rat transient receptor potential vanilloid 1 receptor (n=2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50163235(4-o-Tolyl-piperidine-1-carboxylic acid (4-trifluor...)
Affinity DataEC50:  1.72E+3nMAssay Description:Effective concentration against rat transient receptor potential vanilloid 1 receptor (n=2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50130539(2,2-Dimethyl-propionic acid 2-(3,4-dimethyl-benzyl...)
Affinity DataEC50:  790nMAssay Description:In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50130544(Benzoic acid 2-(4-tert-butyl-benzyl)-3-[3-(4-metha...)
Affinity DataEC50:  252nMAssay Description:In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50130545(Benzoic acid 2-(4-tert-butyl-benzyl)-3-[3-(4-metha...)
Affinity DataEC50:  2.79E+3nMAssay Description:In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50130548(2,2-Dimethyl-propionic acid 2-(3,4-dimethyl-benzyl...)
Affinity DataEC50:  22nMAssay Description:In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50130538(2,2-Dimethyl-propionic acid 3-[3-(4-acetylamino-be...)
Affinity DataEC50:  450nMAssay Description:In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50130546(2,2-Dimethyl-propionic acid 2-(4-tert-butyl-benzyl...)
Affinity DataEC50:  40nMAssay Description:In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50130552(Benzoic acid 2-(3,4-dimethyl-benzyl)-3-[3-(4-metha...)
Affinity DataEC50:  166nMAssay Description:In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50130551(2,2-Dimethyl-propionic acid 2-(3,4-dimethyl-benzyl...)
Affinity DataEC50:  1.70E+3nMAssay Description:In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50196337(2-((3-(4-hydroxy-3-methoxybenzyl)thioureido)methyl...)
Affinity DataEC50:  1.97nMAssay Description:In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50196343(2-((3-(4-hydroxy-3-methoxybenzyl)thioureido)methyl...)
Affinity DataEC50:  2.83nMAssay Description:In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM20461(Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...)
Affinity DataEC50:  44.8nMAssay Description:In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50130556(Benzoic acid 2-(3,4-dimethyl-benzyl)-3-[3-(4-metha...)
Affinity DataEC50:  1.73E+3nMAssay Description:In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50130554(2,2-Dimethyl-propionic acid 2-(3,4-dimethyl-benzyl...)
Affinity DataEC50:  1.14E+3nMAssay Description:In vitro [Ca2+] influx relative to capsaicin by Rat Vanilloid receptor (VR1) expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Displayed 1 to 50 (of 2928 total ) | Next | Last >>
Jump to: