Compile Data Set for Download or QSAR
Report error Found 92 of affinity data for UniProtKB/TrEMBL: O19045
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50266924((2R,4S)-N1-(4-Chlorophenyl)-4-(2,4-difluorophenyl)...)
Affinity DataIC50: 0.108nMAssay Description:Inhibition of rabbit F10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM17283((2S)-3-(7-carbamimidoylnaphthalen-2-yl)-2-(4-{[(3S...)
Affinity DataIC50: 41nMAssay Description:Compound was tested for the inhibition of serine protease factor Xa enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080132(CHEMBL3415976)
Affinity DataIC50: 460nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM7840(RIVAROXABAN | US8822458, 97 | US8822458, 44)
Affinity DataIC50: 510nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080107(CHEMBL3415998)
Affinity DataIC50: 720nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080132(CHEMBL3415976)
Affinity DataIC50: 750nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080131(CHEMBL3415975)
Affinity DataIC50: 780nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080133(CHEMBL3415977)
Affinity DataIC50: 810nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080143(CHEMBL3415984)
Affinity DataIC50: 820nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM7840(RIVAROXABAN | US8822458, 97 | US8822458, 44)
Affinity DataIC50: 860nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080101(CHEMBL3415997)
Affinity DataIC50: 890nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080142(CHEMBL3415983)
Affinity DataIC50: 910nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080100(CHEMBL3415996)
Affinity DataIC50: 920nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080107(CHEMBL3415998)
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080143(CHEMBL3415984)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080101(CHEMBL3415997)
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080100(CHEMBL3415996)
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080131(CHEMBL3415975)
Affinity DataIC50: 1.39E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080133(CHEMBL3415977)
Affinity DataIC50: 1.52E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080134(CHEMBL3415978)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080142(CHEMBL3415983)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080099(CHEMBL3415995)
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080078(CHEMBL3415987)
Affinity DataIC50: 1.78E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080099(CHEMBL3415995)
Affinity DataIC50: 1.91E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080078(CHEMBL3415987)
Affinity DataIC50: 1.96E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080077(CHEMBL3415986)
Affinity DataIC50: 1.98E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080134(CHEMBL3415978)
Affinity DataIC50: 1.98E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080096(CHEMBL3415985)
Affinity DataIC50: 2.45E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080077(CHEMBL3415986)
Affinity DataIC50: 2.56E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080126(CHEMBL3415999)
Affinity DataIC50: 2.78E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080135(CHEMBL3415979)
Affinity DataIC50: 2.89E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080079(CHEMBL3415988)
Affinity DataIC50: 2.98E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080096(CHEMBL3415985)
Affinity DataIC50: 3.01E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080126(CHEMBL3415999)
Affinity DataIC50: 3.04E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080127(CHEMBL3416000)
Affinity DataIC50: 3.12E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080136(CHEMBL3415980)
Affinity DataIC50: 3.19E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080135(CHEMBL3415979)
Affinity DataIC50: 3.23E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080137(CHEMBL3415981)
Affinity DataIC50: 3.45E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080127(CHEMBL3416000)
Affinity DataIC50: 3.46E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080136(CHEMBL3415980)
Affinity DataIC50: 3.52E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080079(CHEMBL3415988)
Affinity DataIC50: 3.67E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080137(CHEMBL3415981)
Affinity DataIC50: 3.78E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080128(CHEMBL3416001)
Affinity DataIC50: 3.78E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080141(CHEMBL3415982)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080128(CHEMBL3416001)
Affinity DataIC50: 4.02E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080130(CHEMBL3416003)
Affinity DataIC50: 4.06E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080141(CHEMBL3415982)
Affinity DataIC50: 4.14E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080129(CHEMBL3416002)
Affinity DataIC50: 4.23E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of prothombin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080130(CHEMBL3416003)
Affinity DataIC50: 4.79E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetCoagulation factor X(Rabbit)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50080129(CHEMBL3416002)
Affinity DataIC50: 5.12E+3nMAssay Description:Inhibition of F10a in rabbit plasma assessed as doubling of activated partial thromboplastin timeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
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