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Report error Found 625 for UniProtKB: O15151
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM35084(N-acylpolyamine (NAPA) scaffold, 35)
Affinity DataAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2009
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50327206((2S,5S,8S,11S,14S,17S,20S,23S,26S,29S)-11-((1H-ind...)
Affinity DataKd:  390nMAssay Description:Binding affinity to MDMXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50261655(CHEMBL4090785)
Affinity DataKd:  21nMAssay Description:Inhibition of p53 binding to MDMX (unknown origin) after 30 mins by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50261654(CHEMBL4076935)
Affinity DataKd:  84nMAssay Description:Inhibition of p53 binding to MDMX (unknown origin) after 30 mins by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50261658(CHEMBL4099164)
Affinity DataKd:  61nMAssay Description:Inhibition of p53 binding to MDMX (unknown origin) after 30 mins by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50261659(CHEMBL4059725)
Affinity DataKd:  614nMAssay Description:Inhibition of p53 binding to MDMX (unknown origin) after 30 mins by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50261656(CHEMBL3347578)
Affinity DataKd:  8.5nMAssay Description:Inhibition of p53 binding to MDMX (unknown origin) after 30 mins by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50261657(CHEMBL4075572)
Affinity DataKd:  19nMAssay Description:Inhibition of p53 binding to MDMX (unknown origin) after 30 mins by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2020
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50287913(CHEMBL4175039)
Affinity DataKd:  2.30nMAssay Description:Binding affinity to full length human MDM4 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2020
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50506487(CHEMBL4441886)
Affinity DataKd:  221nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50506484(CHEMBL4530683)
Affinity DataKd:  641nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50506489(CHEMBL4592815)
Affinity DataKd:  440nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50506485(CHEMBL4460980)
Affinity DataKd:  279nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50506491(CHEMBL4521951)
Affinity DataKd:  370nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50506490(CHEMBL4460091)
Affinity DataKd:  593nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50014089(CHEMBL1236726)
Affinity DataEC50:  2.00E+4nMAssay Description:Inhibition of p53 protein binding to MDMX (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50554653(CHEMBL4750962)
Affinity DataKd:  67nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50554654(CHEMBL4799193)
Affinity DataKd:  187nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50554655(CHEMBL4795544)
Affinity DataKd:  781nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50554656(CHEMBL4741500)
Affinity DataKd:  251nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50554657(CHEMBL4778122)
Affinity DataKd:  372nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50554658(CHEMBL4786907)
Affinity DataKd:  265nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50554659(CHEMBL4763522)
Affinity DataKd:  242nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50554661(CHEMBL4800669)
Affinity DataKd:  115nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50554662(CHEMBL4799966)
Affinity DataKd:  348nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50554663(CHEMBL4785105)
Affinity DataKd:  1.68E+3nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50554664(CHEMBL4789508)
Affinity DataKd:  570nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50590814(CHEMBL5182359)
Affinity DataKd:  27nMAssay Description:Binding affinity to N-terminal TEV/GST-fused human MDM4 (22 to 110 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation consta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50624183(CHEMBL5394570)
Affinity DataKd:  6.90nMAssay Description:Binding affinity to 6x-His-TEV-tagged human MDMX (15 to 111 residues) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50624184(CHEMBL5415331)
Affinity DataKd:  57nMAssay Description:Binding affinity to 6x-His-TEV-tagged human MDMX (15 to 111 residues) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50624185(CHEMBL5439046)
Affinity DataKd:  7nMAssay Description:Binding affinity to 6x-His-TEV-tagged human MDMX (15 to 111 residues) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50403301(CHEMBL4289676)
Affinity DataKd:  210nMAssay Description:Binding affinity to human MDM4 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50403305(CHEMBL5275075)
Affinity DataKd:  229nMAssay Description:Binding affinity to human MDM4 assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50403306(CHEMBL5271788)
Affinity DataKd:  13nMAssay Description:Binding affinity to human MDM4 assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50403367(CHEMBL5283428)
Affinity DataKd:  25nMAssay Description:Binding affinity to human MDM4 assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50403367(CHEMBL5283428)
Affinity DataKd:  43nMAssay Description:Binding affinity to human MDM4 assessed as dissociation constant by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50403526(CHEMBL5286722)
Affinity DataEC50:  2.30E+3nMAssay Description:Inhibition of human MDM4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50403527(CHEMBL5280949)
Affinity DataKd:  27nMAssay Description:Inhibition of human his-tagged MDM4 assessed as dissociation constant by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50437206(CHEMBL2402737 | US20250073340, Example RG7388)
Affinity DataKd: <100nMAssay Description:Inhibition of MDM4 assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50646908(CHEMBL5593887)
Affinity DataKd:  8.20E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50646909(CHEMBL5593552)
Affinity DataKd:  7.70E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50646910(CHEMBL5592519)
Affinity DataKd:  1.14E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50646911(CHEMBL5593173)
Affinity DataKd:  6.46E+5nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50646912(CHEMBL5594551)
Affinity DataKd:  1.29E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50646913(CHEMBL5583823)
Affinity DataKd:  2.47E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50646914(CHEMBL5590250)
Affinity DataKd:  1.09E+5nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50646915(CHEMBL5595494)
Affinity DataKd:  7.00E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50646916(CHEMBL5595333)
Affinity DataKd:  2.47E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50646917(CHEMBL5593177)
Affinity DataKd:  1.09E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein Mdm4(Human)
Nih

LigandPNGBDBM50014089(CHEMBL1236726)
Affinity DataKd:  1.10E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
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