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Report error Found 18 for UniProtKB: O00560
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50632490(CHEMBL5439384)
Affinity DataKd:  1.80E+3nMAssay Description:Binding affinity to full length N-terminal GST-tagged human syntenin-1 expressed in Escherichia coli ER2566 assessed as dissociation constant by ITC ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetSyndecan-2/Syntenin-1(Human)
Aix-Marseille Universit£

Curated by ChEMBL
LigandPNGBDBM50574543(CHEMBL4874274)
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of recombinant human full-length GST-tagged syntenin-1/Syndecan-2 complex interaction expressed in Escherichia coli ER2566 measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50557298(CHEMBL4750927)
Affinity DataKi:  30nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50557293(CHEMBL4781637)
Affinity DataKi:  40nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50557299(CHEMBL4799812)
Affinity DataKi:  170nMAssay Description:Binding affinity to syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50557299(CHEMBL4799812)
Affinity DataKi:  190nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50557294(CHEMBL4749490)
Affinity DataKi:  250nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50557297(CHEMBL4747962)
Affinity DataKi:  250nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50557296(CHEMBL4792861)
Affinity DataKi:  250nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50557295(CHEMBL4758599)
Affinity DataKi:  250nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50557287(CHEMBL4752622)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50557286(CHEMBL4798461)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50557288(CHEMBL4792781)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50557289(CHEMBL4740875)
Affinity DataKi:  2.40E+4nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50557290(CHEMBL4798840)
Affinity DataKi:  4.40E+4nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50557291(CHEMBL4785814)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50557292(CHEMBL4779632)
Affinity DataKi:  1.10E+5nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSyntenin-1(Human)
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50557285(CHEMBL4788058)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of syntenin-PDZ1-2 domain (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 5 mins by fluorescence polarization assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed