LigandBDBM254266(US9464084, 158 | US10112937, Example 158 | US10150...)
Affinity DataIC50: 7.90nMAssay Description:Antagonist activity at macaque P2X7 assessed as inhibition of BzATP-induced calcium flux preincubated for 30 mins followed by BzATP addition measured...More data for this Ligand-Target Pair