Compile Data Set for Download or QSAR
Report error Found 8 of affinity data for UniProtKB/TrEMBL: C5ISA2
TargetTubulin alpha chain(Sheep)TBA
LigandPNGBDBM50487731(CHEMBL2262117)
Affinity DataKd:  3.70E+3nMAssay Description:Binding affinity to Ovis aries (sheep) brain tubulin assessed as intrinsic tryptophan fluorescence after 30 min by fluorescence spectroscopic analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetTubulin alpha chain(Sheep)TBA
LigandPNGBDBM50487731(CHEMBL2262117)
Affinity DataIC50: 1.96E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 30 min by CD spectra analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetTubulin alpha chain(Sheep)TBA
LigandPNGBDBM50487731(CHEMBL2262117)
Affinity DataIC50: 1.96E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetTubulin alpha chain(Sheep)TBA
LigandPNGBDBM86012(Chalcone, 11)
Affinity DataIC50: 2.03E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetTubulin alpha chain(Sheep)TBA
LigandPNGBDBM50487732(CHEMBL2262305)
Affinity DataIC50: 2.14E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetTubulin alpha chain(Sheep)TBA
LigandPNGBDBM50067040(CHEMBL116438 | 1,7-bis(4-hydroxy-3-methoxyphenyl)1...)
Affinity DataIC50: 2.66E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetTubulin alpha chain(Sheep)TBA
LigandPNGBDBM86007(Chalcone, 6)
Affinity DataIC50: 4.93E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetTubulin alpha chain(Sheep)TBA
LigandPNGBDBM50487733(CHEMBL2262116)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Ovis aries (sheep) brain tubulin polymerization assessed as microtubule assembly after 15 min by measuring turbidity based spectroscopi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article