Compile Data Set for Download or QSAR
Report error Found 82 of affinity data for UniProtKB/TrEMBL: A5Z252
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(CHEBI:85202 | BCX-1812 | Peramivir)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase expressed in HEK293 cells pre-incubated for 10 mins before 4-M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of Influenza A virus (A/chicken/Bangli/BBVD-563/2007(H5N1)) clade 2 neuraminidase activity using 4-MUNANA as substrate preincubated for 60...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of Influenza A virus (A/Turkey/651242/2006(H5N1)) neuraminidase by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028516(CHEMBL3342478)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028523(CHEMBL3342485)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50464877(CHEMBL4288789)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase expressed in HEK293 cells pre-incubated for 10 mins before 4-M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028511(CHEMBL3342474)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50464876(CHEMBL4288995)
Affinity DataIC50: 4nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase expressed in HEK293 cells pre-incubated for 10 mins before 4-M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028503(Guanidino-Oseltamivir Carboxylicacid | CHEMBL81717)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028508(CHEMBL3342471)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of Influenza A virus A/Anhui/1/2005(H5N1) neuraminidase N1 H274Y mutant using fluorogenic MUNANA as substrate preincubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50464877(CHEMBL4288789)
Affinity DataIC50: 10nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase H275Y mutant expressed in HEK293 cells pre-incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028513(CHEMBL3342476)
Affinity DataIC50: 10nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 11nMAssay Description:Inhibition of Influenza A virus (A/chicken/Bangli/BBVD-563/2007(H5N1)) clade 2 neuraminidase activity using 4-MUNANA as substrate measured every min ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028521(CHEMBL3342483)
Affinity DataIC50: 11nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 11nMAssay Description:Inhibition of Influenza A virus (A/Turkey/651242/2006(H5N1)) neuraminidase by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028512(CHEMBL3342475)
Affinity DataIC50: 13nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028514(CHEMBL3342477)
Affinity DataIC50: 14nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028507(CHEMBL3342470)
Affinity DataIC50: 15nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM5025(ethyl (3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-y...)
Affinity DataIC50: 17nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(CHEBI:85202 | BCX-1812 | Peramivir)
Affinity DataIC50: 18nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase H275Y mutant expressed in HEK293 cells pre-incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028505(CHEMBL3342468)
Affinity DataIC50: 19nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028510(CHEMBL3342473)
Affinity DataIC50: 21nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028525(CHEMBL3355596)
Affinity DataIC50: 21nMAssay Description:Inhibition of Influenza A virus H1N1 Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028525(CHEMBL3355596)
Affinity DataIC50: 25nMAssay Description:Inhibition of Influenza A virus H3N2 Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028504(CHEMBL3342467)
Affinity DataIC50: 27nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028509(CHEMBL3342472)
Affinity DataIC50: 31nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028517(CHEMBL3342479)
Affinity DataIC50: 32nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50469488(CHEMBL4287425)
Affinity DataIC50: 33nMAssay Description:Inhibition of Influenza A virus A/Anhui/1/2005(H5N1) neuraminidase N1 H274Y mutant using fluorogenic MUNANA as substrate preincubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50469486(CHEMBL4276773)
Affinity DataIC50: 36nMAssay Description:Inhibition of Influenza A virus A/Anhui/1/2005(H5N1) neuraminidase N1 H274Y mutant using fluorogenic MUNANA as substrate preincubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028522(CHEMBL3342484)
Affinity DataIC50: 43nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028519(CHEMBL3342481)
Affinity DataIC50: 59nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50464876(CHEMBL4288995)
Affinity DataIC50: 73nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase H275Y mutant expressed in HEK293 cells pre-incubated for 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028506(CHEMBL3342469)
Affinity DataIC50: 78nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028520(CHEMBL3342482)
Affinity DataIC50: 90nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028483(CHEMBL3342331)
Affinity DataIC50: 100nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028482(CHEMBL3342330)
Affinity DataIC50: 100nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028518(CHEMBL3342480)
Affinity DataIC50: 100nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028490(CHEMBL3342459)
Affinity DataIC50: 150nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50464469(CHEMBL4280059)
Affinity DataIC50: 190nMAssay Description:Inhibition of Influenza A virus A/Anhui/1/2005(H5N1) neuraminidase using MUNANA as substrate preincubated for 5 to 15 mins followed by substrate addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028484(CHEMBL3342456)
Affinity DataIC50: 200nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM5025(ethyl (3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-y...)
Affinity DataIC50: 210nMAssay Description:Inhibition of Influenza A virus A/Anhui/1/2005(H5N1) neuraminidase using MUNANA as substrate preincubated for 5 to 15 mins followed by substrate addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50464464(CHEMBL4287286)
Affinity DataIC50: 228nMAssay Description:Inhibition of Influenza A virus A/Anhui/1/2005(H5N1) neuraminidase using MUNANA as substrate preincubated for 5 to 15 mins followed by substrate addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028497(CHEMBL3342461)
Affinity DataIC50: 230nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50464466(CHEMBL4295229)
Affinity DataIC50: 238nMAssay Description:Inhibition of Influenza A virus A/Anhui/1/2005(H5N1) neuraminidase using MUNANA as substrate preincubated for 5 to 15 mins followed by substrate addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50464463(CHEMBL4290699)
Affinity DataIC50: 266nMAssay Description:Inhibition of Influenza A virus A/Anhui/1/2005(H5N1) neuraminidase using MUNANA as substrate preincubated for 5 to 15 mins followed by substrate addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50271273(CHEMBL4127125)
Affinity DataIC50: 281nMAssay Description:Inhibition of Influenza A virus (A/chicken/Bangli/BBVD-563/2007(H5N1)) clade 2 neuraminidase activity using 4-MUNANA as substrate measured every min ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50271273(CHEMBL4127125)
Affinity DataIC50: 316nMAssay Description:Inhibition of Influenza A virus (A/chicken/Bangli/BBVD-563/2007(H5N1)) clade 2 neuraminidase activity using 4-MUNANA as substrate preincubated for 60...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50469490(CHEMBL4282553)
Affinity DataIC50: 364nMAssay Description:Inhibition of Influenza A virus A/Anhui/1/2005(H5N1) neuraminidase N1 H274Y mutant using fluorogenic MUNANA as substrate preincubated for 10 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50028500(CHEMBL3342464)
Affinity DataIC50: 370nMAssay Description:Inhibition of Influenza A virus A/chicken/china/1220/2012(H5N1) Neuraminidase N1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2016
Entry Details Article
PubMed
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