Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 1773
TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandPNGBDBM200747(US9233108, 9 | US9757383, Example 9)
Affinity DataIC50: 0.200nMAssay Description:The study of binding to human muscarinic M1, M2, M3, M4 and M5 receptors was performed using commercial membranes (Perkin Elmer) prepared from CHO-K1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandPNGBDBM200741(US9233108, 1 | US9757383, Example 1)
Affinity DataIC50: 0.300nMAssay Description:The study of binding to human muscarinic M1, M2, M3, M4 and M5 receptors was performed using commercial membranes (Perkin Elmer) prepared from CHO-K1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandPNGBDBM200748(US9233108, 10 | US9757383, Example 10)
Affinity DataIC50: 0.400nMAssay Description:The study of binding to human muscarinic M1, M2, M3, M4 and M5 receptors was performed using commercial membranes (Perkin Elmer) prepared from CHO-K1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandPNGBDBM200753(US9233108, 18 | US9757383, Example 18)
Affinity DataIC50: 0.400nMAssay Description:The study of binding to human muscarinic M1, M2, M3, M4 and M5 receptors was performed using commercial membranes (Perkin Elmer) prepared from CHO-K1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandPNGBDBM200744(US9233108, 5 | US9757383, Example 5)
Affinity DataIC50: 0.400nMAssay Description:The study of binding to human muscarinic M1, M2, M3, M4 and M5 receptors was performed using commercial membranes (Perkin Elmer) prepared from CHO-K1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandPNGBDBM200742(US9233108, 2 | US9757383, Example 2)
Affinity DataIC50: 0.400nMAssay Description:The study of binding to human muscarinic M1, M2, M3, M4 and M5 receptors was performed using commercial membranes (Perkin Elmer) prepared from CHO-K1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandPNGBDBM200749(US9233108, 11 | US9757383, Example 11)
Affinity DataIC50: 0.5nMAssay Description:The study of binding to human muscarinic M1, M2, M3, M4 and M5 receptors was performed using commercial membranes (Perkin Elmer) prepared from CHO-K1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandPNGBDBM339881(US9757383, Example 4 | trans-4-[{3-[5-({[(2R)-2-hy...)
Affinity DataIC50: 0.600nMAssay Description:The study of binding to human muscarinic M1, M2, M3, M4 and M5 receptors was performed using commercial membranes (Perkin Elmer) prepared from CHO-K1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandPNGBDBM339892(US9757383, Example 17 | trans-4-[{3-[5-({[(2R)-2-h...)
Affinity DataIC50: 0.600nMAssay Description:The study of binding to human muscarinic M1, M2, M3, M4 and M5 receptors was performed using commercial membranes (Perkin Elmer) prepared from CHO-K1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandPNGBDBM200754(US9233108, 19 | US9757383, Example 19)
Affinity DataIC50: 0.800nMAssay Description:The study of binding to human muscarinic M1, M2, M3, M4 and M5 receptors was performed using commercial membranes (Perkin Elmer) prepared from CHO-K1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandPNGBDBM200750(US9233108, 15 | US9757383, Example 15)
Affinity DataIC50: 1nMAssay Description:The study of binding to human muscarinic M1, M2, M3, M4 and M5 receptors was performed using commercial membranes (Perkin Elmer) prepared from CHO-K1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetBeta-2 adrenergic receptor(Human)
Almirall

US Patent
LigandPNGBDBM200753(US9233108, 18 | US9757383, Example 18)
Affinity DataIC50: 1.40nMAssay Description:The study of binding to human adrenergic beta1 and beta2 receptors was performed using commercial membranes prepared from Sf9 cells where they are ov...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandPNGBDBM339883(US9757383, Example 6 | trans-4-[{2-[{[4-({[(2R)-2-...)
Affinity DataIC50: 1.40nMAssay Description:The study of binding to human muscarinic M1, M2, M3, M4 and M5 receptors was performed using commercial membranes (Perkin Elmer) prepared from CHO-K1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetBeta-2 adrenergic receptor(Human)
Almirall

US Patent
LigandPNGBDBM200750(US9233108, 15 | US9757383, Example 15)
Affinity DataIC50: 1.5nMAssay Description:The study of binding to human adrenergic beta1 and beta2 receptors was performed using commercial membranes prepared from Sf9 cells where they are ov...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
Go to US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandPNGBDBM200746(US9233108, 8 | US9757383, Example 8)
Affinity DataIC50: 2.20nMAssay Description:The study of binding to human muscarinic M1, M2, M3, M4 and M5 receptors was performed using commercial membranes (Perkin Elmer) prepared from CHO-K1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetBeta-2 adrenergic receptor(Human)
Almirall

US Patent
LigandPNGBDBM200747(US9233108, 9 | US9757383, Example 9)
Affinity DataIC50: 2.20nMAssay Description:The study of binding to human adrenergic beta1 and beta2 receptors was performed using commercial membranes prepared from Sf9 cells where they are ov...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
Go to US Patent

TargetBeta-2 adrenergic receptor(Human)
Almirall

US Patent
LigandPNGBDBM200744(US9233108, 5 | US9757383, Example 5)
Affinity DataIC50: 2.70nMAssay Description:The study of binding to human adrenergic beta1 and beta2 receptors was performed using commercial membranes prepared from Sf9 cells where they are ov...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetBeta-2 adrenergic receptor(Human)
Almirall

US Patent
LigandPNGBDBM200755(US9233108, 20 | US9757383, Example 20)
Affinity DataIC50: 3.10nMAssay Description:The study of binding to human adrenergic beta1 and beta2 receptors was performed using commercial membranes prepared from Sf9 cells where they are ov...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandPNGBDBM200755(US9233108, 20 | US9757383, Example 20)
Affinity DataIC50: 3.60nMAssay Description:The study of binding to human muscarinic M1, M2, M3, M4 and M5 receptors was performed using commercial membranes (Perkin Elmer) prepared from CHO-K1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetBeta-2 adrenergic receptor(Human)
Almirall

US Patent
LigandPNGBDBM200749(US9233108, 11 | US9757383, Example 11)
Affinity DataIC50: 4.20nMAssay Description:The study of binding to human adrenergic beta1 and beta2 receptors was performed using commercial membranes prepared from Sf9 cells where they are ov...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
Go to US Patent

TargetBeta-2 adrenergic receptor(Human)
Almirall

US Patent
LigandPNGBDBM200748(US9233108, 10 | US9757383, Example 10)
Affinity DataIC50: 5.70nMAssay Description:The study of binding to human adrenergic beta1 and beta2 receptors was performed using commercial membranes prepared from Sf9 cells where they are ov...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
Go to US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandPNGBDBM200752(US9233108, 17 | US9757383, Example 16)
Affinity DataIC50: 5.90nMAssay Description:The study of binding to human muscarinic M1, M2, M3, M4 and M5 receptors was performed using commercial membranes (Perkin Elmer) prepared from CHO-K1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetBeta-2 adrenergic receptor(Human)
Almirall

US Patent
LigandPNGBDBM200752(US9233108, 17 | US9757383, Example 16)
Affinity DataIC50: 12nMAssay Description:The study of binding to human adrenergic beta1 and beta2 receptors was performed using commercial membranes prepared from Sf9 cells where they are ov...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
Go to US Patent

TargetBeta-2 adrenergic receptor(Human)
Almirall

US Patent
LigandPNGBDBM339892(US9757383, Example 17 | trans-4-[{3-[5-({[(2R)-2-h...)
Affinity DataIC50: 13nMAssay Description:The study of binding to human adrenergic beta1 and beta2 receptors was performed using commercial membranes prepared from Sf9 cells where they are ov...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
Go to US Patent

TargetBeta-2 adrenergic receptor(Human)
Almirall

US Patent
LigandPNGBDBM200746(US9233108, 8 | US9757383, Example 8)
Affinity DataIC50: 18nMAssay Description:The study of binding to human adrenergic beta1 and beta2 receptors was performed using commercial membranes prepared from Sf9 cells where they are ov...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
Go to US Patent

TargetBeta-2 adrenergic receptor(Human)
Almirall

US Patent
LigandPNGBDBM339883(US9757383, Example 6 | trans-4-[{2-[{[4-({[(2R)-2-...)
Affinity DataIC50: 34nMAssay Description:The study of binding to human adrenergic beta1 and beta2 receptors was performed using commercial membranes prepared from Sf9 cells where they are ov...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
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TargetBeta-2 adrenergic receptor(Human)
Almirall

US Patent
LigandPNGBDBM200754(US9233108, 19 | US9757383, Example 19)
Affinity DataIC50: 62nMAssay Description:The study of binding to human adrenergic beta1 and beta2 receptors was performed using commercial membranes prepared from Sf9 cells where they are ov...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
Go to US Patent

TargetBeta-2 adrenergic receptor(Human)
Almirall

US Patent
LigandPNGBDBM200742(US9233108, 2 | US9757383, Example 2)
Affinity DataIC50: 120nMAssay Description:The study of binding to human adrenergic beta1 and beta2 receptors was performed using commercial membranes prepared from Sf9 cells where they are ov...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
Go to US Patent

TargetBeta-2 adrenergic receptor(Human)
Almirall

US Patent
LigandPNGBDBM200741(US9233108, 1 | US9757383, Example 1)
Affinity DataIC50: 140nMAssay Description:The study of binding to human adrenergic beta1 and beta2 receptors was performed using commercial membranes prepared from Sf9 cells where they are ov...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
Go to US Patent

TargetBeta-2 adrenergic receptor(Human)
Almirall

US Patent
LigandPNGBDBM339881(US9757383, Example 4 | trans-4-[{3-[5-({[(2R)-2-hy...)
Affinity DataIC50: 220nMAssay Description:The study of binding to human adrenergic beta1 and beta2 receptors was performed using commercial membranes prepared from Sf9 cells where they are ov...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details
Go to US Patent