Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 6920
TargetBeta-lactamase(Escherichia coli (strain K12))
Meiji Seika Pharma

US Patent
LigandPNGBDBM159600(US9035062, 23 | US8772490, Example 23)
Affinity DataIC50: 650nMpH: 7.0Assay Description:For the measurement of β-lactamase inhibitory activity, 100 μM (final concentration) nitrocefin (Oxoid) was used as a substrate, and 2.5% D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2015
Entry Details
Go to US Patent

TargetBeta-lactamase(Escherichia coli (strain K12))
Meiji Seika Pharma

US Patent
LigandPNGBDBM50157692(CHEMBL1439 | Sodium; (2S,3S,5R)-3-methyl-4,4,7-tri...)
Affinity DataIC50: 950nMpH: 7.0Assay Description:For the measurement of β-lactamase inhibitory activity, 100 μM (final concentration) nitrocefin (Oxoid) was used as a substrate, and 2.5% D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2015
Entry Details
Go to US Patent

TargetBeta-lactamase(Escherichia coli (strain K12))
Meiji Seika Pharma

US Patent
LigandPNGBDBM159601(US9035062, 24 | US8772490, Example 24)
Affinity DataIC50: 3.00E+4nMpH: 7.0Assay Description:For the measurement of β-lactamase inhibitory activity, 100 μM (final concentration) nitrocefin (Oxoid) was used as a substrate, and 2.5% D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2015
Entry Details
Go to US Patent