Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 12129
TargetSerine/threonine-protein kinase pim-1(Human)
CNIO

US Patent
LigandPNGBDBM681801(US20240199630, Compound T4.9)
Affinity DataIC50: 0.800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase pim-1(Human)
CNIO

US Patent
LigandPNGBDBM681796(US20240199630, Compound T4.1)
Affinity DataIC50: 0.900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase pim-1(Human)
CNIO

US Patent
LigandPNGBDBM681799(US20240199630, Compound T4.7)
Affinity DataIC50: 1.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase pim-1(Human)
CNIO

US Patent
LigandPNGBDBM681800(US20240199630, Compound T4.8)
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681768(US20240199630, Compound 1)
Affinity DataIC50: 4.80nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681770(US20240199630, Compound 2 | US20240199630, Compoun...)
Affinity DataIC50: 5.03nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase pim-1(Human)
CNIO

US Patent
LigandPNGBDBM681797(US20240199630, Compound T4.2)
Affinity DataIC50: 5.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681783(US20240199630, Compound 34)
Affinity DataIC50: 5.87nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681783(US20240199630, Compound 34)
Affinity DataIC50: 5.87nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681781(US20240199630, Compound 33)
Affinity DataIC50: 6.37nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681781(US20240199630, Compound 33)
Affinity DataIC50: 6.37nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase pim-1(Human)
CNIO

US Patent
LigandPNGBDBM681798(US20240199630, Compound T4.6)
Affinity DataIC50: 8.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681772(US20240199630, Compound 3 | US20240199630, Compoun...)
Affinity DataIC50: 10.2nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681785(US20240199630, Compound 35)
Affinity DataIC50: 20.7nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681785(US20240199630, Compound 35)
Affinity DataIC50: 20.7nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681773(US20240199630, Compound 25)
Affinity DataIC50: 22.3nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681774(US20240199630, Compound 4 | US20240199630, Compoun...)
Affinity DataIC50: 24.7nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681776(US20240199630, Compound 5)
Affinity DataIC50: 36.5nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681780(US20240199630, Compound 7)
Affinity DataIC50: 40.2nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681782(US20240199630, Compound 10 | US20240199630, Compou...)
Affinity DataIC50: 50.5nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681778(US20240199630, Compound 6)
Affinity DataIC50: 53.2nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681784(US20240199630, Compound 12 | US20240199630, Compou...)
Affinity DataIC50: 61.3nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681786(US20240199630, Compound 13)
Affinity DataIC50: 69.8nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681775(US20240199630, Compound 27)
Affinity DataIC50: 75.2nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681777(US20240199630, Compound 28)
Affinity DataIC50: 101nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681787(US20240199630, Compound 14)
Affinity DataIC50: 133nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681788(US20240199630, Compound 15)
Affinity DataIC50: 145nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681779(US20240199630, Compound 31)
Affinity DataIC50: 221nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681769(US20240199630, Compound 17)
Affinity DataIC50: 225nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase haspin(Human)
CNIO

US Patent
LigandPNGBDBM681771(US20240199630, Compound 18)
Affinity DataIC50: 231nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase pim-1(Human)
CNIO

US Patent
LigandPNGBDBM681782(US20240199630, Compound 10 | US20240199630, Compou...)
Affinity DataIC50: 1.09E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase pim-1(Human)
CNIO

US Patent
LigandPNGBDBM681784(US20240199630, Compound 12 | US20240199630, Compou...)
Affinity DataIC50: 1.81E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase pim-1(Human)
CNIO

US Patent
LigandPNGBDBM681774(US20240199630, Compound 4 | US20240199630, Compoun...)
Affinity DataIC50: 2.27E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase pim-1(Human)
CNIO

US Patent
LigandPNGBDBM681795(US20240199630, Compound T3.27)
Affinity DataIC50: 3.18E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase pim-1(Human)
CNIO

US Patent
LigandPNGBDBM681792(US20240199630, Compound T3.6)
Affinity DataIC50: 3.30E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase pim-1(Human)
CNIO

US Patent
LigandPNGBDBM681770(US20240199630, Compound 2 | US20240199630, Compoun...)
Affinity DataIC50: 3.40E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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TargetSerine/threonine-protein kinase pim-1(Human)
CNIO

US Patent
LigandPNGBDBM681772(US20240199630, Compound 3 | US20240199630, Compoun...)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
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