Compile Data Set for Download or QSAR
Report error Found 172 Enz. Inhib. hit(s) with all data for entry = 10322
TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438838(US10604489, Compound 2 | US11180455, Compound 2)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438839(3-((1R,5S,9r)-9-methoxy-3-(2-oxaspiro[3.5]nonan-7-...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438841(3-((1R,5S,9r)-9-methoxy-3-(7-oxaspiro[3.5]nonan-2-...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438844(3-((1R,5S,9r)-3-(4,4-difluorocyclohexyl)-9-methoxy...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438846(3-((1R,5S,9r)-3-(bicyclo[3.1.0]hexan-3-yl)-9-metho...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438845(US10604489, Compound 10 | US11180455, Compound 202)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438849(4-((1R,5S,9r)-9-methoxy-3-(7-oxaspiro[3.5]nonan-2-...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438850(US10604489, Compound 14 | US11180455, Compound 203)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438853(3-((1R,5S,9R)-3-((1R,3r,5S)-6,6-difluorobicyclo[3....)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438854(4-((1R,5S,9R)-3-((1R,3r,5S)-6,6-difluorobicyclo[3....)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438855(US10604489, Compound 19 | US11180455, Compound 19)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438858(3-((1R,5S,9r)-3-benzyl-9-methoxy-3-azabicyclo[3.3....)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438859(3-((1R,5S,9r)-9-methoxy-3-azabicyclo[3.3.1]nonan-9...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438861(US10604489, Compound 54 | 3-((1R,5S,9r)-9-methoxy-...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438862(3-((1R,5S,9r)-9-methoxy-3-phenethyl-3-azabicyclo[3...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438863(3-((1R,5S,9r)-3-isopropyl-9-methoxy-3-azabicyclo[3...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438864(3-benzyl-1,5,3-dioxazepane | US10604489, Compound ...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438867(3-((1R,5S,9r)-3-butyl-9-methoxy-3-azabicyclo[3.3.1...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438868((1R,5S,9r)-3-(cyclopropylmethyl)-9-ethoxy-9-(3-iod...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438872(3-((1R,5S,9r)-9-methoxy-3-(3,3,3-trifluoropropyl)-...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438873((1R,5S,9r)-tert-butyl 9-(3-hydroxphenyl)-9-methoxy...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438874(5-((1R,5S,9r)-3-(cyclopropylmethyl)-9-methoxy-3-az...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438876(3-((1R,5S,9r)-3-cyclopropyl-9-methoxy-3-azabicyclo...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438878(3-((1R,5S,9r)-3-((1-fluorocyclopropyl)methyl)-9-me...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438880(3-((1R,5S,9r)-3-cyclobutyl-9-methoxy-3-azabicyclo[...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
Go to US Patent

TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438881(4-((1R,5S,9r)-9-methoxy-3-methyl-3-azabicyclo[3.3....)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438884(1-((tetrahydro-2H-pyran-2-yl)oxy)cyclopropanecarbo...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438885(3-((1R,5S,9r)-9-methoxy-3-propyl-3-azabicyclo[3.3....)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438886((1R,5S,9r)-9-(5-bromothiophen-2-yl)-3-methyl-3-aza...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438887(2-hydroxy-3-((1R,5S,9r)-9-methoxy-3-methyl-3-azabi...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438889(3-((1R,5S,9r)-9-methoxy-3-(oxetan-3-ylmethyl)-3-az...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
Go to US Patent

TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438861(US10604489, Compound 54 | 3-((1R,5S,9r)-9-methoxy-...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438893((1R,5S)-3-cyclopentyl-3-azaspiro[bicyclo[3.3.1]non...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438896(3-((1R,5S,9r)-3-((2-hydroxy-2,3-dihydro-1H-inden-2...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
Go to US Patent

TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438902(3-((1R,5S,9r)-9-methoxy-3-(2-(2-oxoimidazolidin-1-...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438903(3-((1R,5S,9r)-3-((1H-benzo[d]imidazol-2-yl)methyl)...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438904(3-((1R,5S,9r)-3-(2-(2,5-dioxopyrrolidin-1-yl)ethyl...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438912(4-((1R,5S,9r)-3-((2-hydroxy-2,3-dihydro-1H-inden-2...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438914(3-((1R,5S,9r)-3-((1H-1,2,3-triazol-5-yl)methyl)-9-...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438916(4-((1R,5S,9r)-9-methoxy-3-(spiro[3.3]heptan-2-yl)-...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438920(4-((1R,5S,9r)-9-methoxy-3-(2-oxaspiro[3.3]heptan-6...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438926(US10604489, Compound 87 | US11180455, Compound 89)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438926(US10604489, Compound 87 | US11180455, Compound 89)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438933(US10604489, Compound 94 | US11180455, Compound 94)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438935(4-((1R,5S,9r)-3-((1H-imidazol-5-yl)methyl)-9-metho...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM528114(US11180455, Compound 97)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438939(4-((1R,5S,9r)-3-((1H-pyrazol-5-yl)methyl)-9-methox...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438941(US10604489, Compound 102 | US11180455, Compound 10...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438943(US10604489, Compound 104 | US11180455, Compound 10...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetMu-type opioid receptor(Human)
TBA

US Patent
LigandPNGBDBM438945(tert-butyl (3-phenylbicyclo[1.1.1]pentan-1-yl)carb...)
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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