Compile Data Set for Download or QSAR
Report error Found 386 Enz. Inhib. hit(s) with all data for entry = 9663
TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480146(rac-(1S,2R)-2-(2-methyl-4- (1-((1-(4-(pyridin-4- y...)
Affinity DataIC50: 3nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480158(rac-(1S,2R)-2-(2-methyl-4- (1-((1-(4-(pyridin-4- y...)
Affinity DataIC50: 3nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480255(rac-(1S,2R)-2-(4-(1-((1-(4- (cyclopropylsulfonyl)p...)
Affinity DataIC50: 3nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480341(rac-(1S,2R)-2-(1-(1-((1-(4- cyanophenyl)azetidin-3...)
Affinity DataIC50: 3nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480343(rac-(1S,2R)-2-(1-(1-((1-(4- cyanophenyl)azetidin-3...)
Affinity DataIC50: 3nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480346(rac-(1S,2R)-2-(1-(3- fluorophenyl)-2-(2-methyl- 1H...)
Affinity DataIC50: 3nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480150(rac-(1S,2R)-2-(2-methyl-4- (1-((1-(4-(pyridin-4- y...)
Affinity DataIC50: 4nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480167(rac-(1S,2R)-2-((1-((1-(4-((4- bromo-1-methyl-1H-py...)
Affinity DataIC50: 4nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480225(rac-N-((1S,2R)-2-(4-(1-((1- (4-((1-methyl-1H-pyraz...)
Affinity DataIC50: 4nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480228(rac-1-((1S,2R)-2-(4-(1-((1- (4- (cyclopropylsulfon...)
Affinity DataIC50: 4nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480260(rac-1-((1S,2R)-2-(2-amino- 1-phenyl-1-(1-((1-(4- (...)
Affinity DataIC50: 4nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480347(rac-(1S,2R)-2-(2-(1H- imidazol-1-yl)-1-(1-((1-(4- ...)
Affinity DataIC50: 4nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480356(rac-(1S,2R)-2-(2-(1H- imidazol-1-yl)-1-phenyl-1- (...)
Affinity DataIC50: 4nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480141(US10899738, Cpd. No 202 | rac-(1S,2R)-2-(2-methyl-...)
Affinity DataIC50: 5nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480210(rac-N-((1S,2R)-2-(2-methyl- 4-(1-((1-(4-(pyridin-4...)
Affinity DataIC50: 5nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480326(rac-(1S,2R)-2-(1-(1-((1-(4- cyanophenyl)azetidin-3...)
Affinity DataIC50: 5nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480342(rac-(1S,2R)-2-(1-(1-((1-(4- chlorophenyl)azetidin-...)
Affinity DataIC50: 5nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50516569(CHEMBL4585198 | US10899738, Cpd. No 148)
Affinity DataIC50: 6nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480099(4-cyclopentyl-2-ethyl-4-(1- ((1-(4-((2-methylpyrid...)
Affinity DataIC50: 6nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480155(rac-(1S,2R)-2- (cyano(phenyl)(1-((1-(4- (pyridin-4...)
Affinity DataIC50: 6nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480291(rac-(1S,2R)-2-((S)- cyano(phenyl)(1-((1-(4- (pyrid...)
Affinity DataIC50: 6nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480314(rac-3-((1S,2R)-2-(2-(1H- imidazol-1-yl)-1-(1-((1-(...)
Affinity DataIC50: 6nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480348(rac-(1S,2R)-2-(1-(1-((1-(4- chlorophenyl)azetidin-...)
Affinity DataIC50: 6nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50516570(CHEMBL4551865 | US10899738, Cpd. No 48)
Affinity DataIC50: 7nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50516571(CHEMBL4592636 | US10899738, Cpd. No 50)
Affinity DataIC50: 7nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480098(4-cyclopentyl-2-ethyl-4-(1- ((1-(4-((3-methylpyrid...)
Affinity DataIC50: 7nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480125(rac-(1S,2R)-2- (cyano(phenyl)(1-((1-(4- (pyridin-4...)
Affinity DataIC50: 7nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480169(rac-(1S,2R)-2-(cyano(1-((1- (4-((1-methyl-1H-pyraz...)
Affinity DataIC50: 7nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480230(rac-1-((1S,2R)-2-(2-ethyl-4- (1-((1-(4-((1-methyl-...)
Affinity DataIC50: 7nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480327(methyl rac-((1S,2R)-2-(2- (1H-imidazol-1-yl)-1-(1-...)
Affinity DataIC50: 7nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480334(methyl rac-((1S,2R)-2-((1- ((1-(4-((4- carbamoylph...)
Affinity DataIC50: 7nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480338(methyl ((1S,2R)-2-((S)- cyano(phenyl)(1-((1-(4- ((...)
Affinity DataIC50: 7nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50516567(CHEMBL4449199 | US10899738, Cpd. No 51)
Affinity DataIC50: 8nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480083(4-cyclopentyl-4-(1-((1-(4- (cyclopropylsulfonyl)ph...)
Affinity DataIC50: 8nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480088(4-cyclopentyl-4-(1-((1-(4- (cyclopentylsulfonyl)ph...)
Affinity DataIC50: 8nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480101(4-cyclopentyl-2-ethyl-4-(1- ((1-(4-((3-ethylpyridi...)
Affinity DataIC50: 8nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480103(4-((4-(3-((4-(4-cyclopentyl- 2-ethyl-1,2,3,4- tetr...)
Affinity DataIC50: 8nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480105(4-((4-(3-((4-(4-cyclopentyl- 2-ethyl-1,2,3,4- tetr...)
Affinity DataIC50: 8nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480177(rac-(1S,2R)-2-(2-(1H- imidazol-1-yl)-1-(1-((1-(4- ...)
Affinity DataIC50: 8nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480216(rac-1-methyl-3-((1S,2R)-2- (2-methyl-4-(1-((1-(4- ...)
Affinity DataIC50: 8nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480300(rac-4-((4-(3-((4-(2-(1H- imidazol-1-yl)-1-((1R,2S)...)
Affinity DataIC50: 8nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480328(methyl rac-((1S,2R)-2- (cyano(phenyl)(1-((1-(4- ((...)
Affinity DataIC50: 8nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50516554(CHEMBL4522767 | US10899738, Cpd. No 49)
Affinity DataIC50: 9nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480082(4-cyclopentyl-2-ethyl-4-(1- ((1-(4- (ethylsulfonyl...)
Affinity DataIC50: 9nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480093(4-cyclopentyl-2-ethyl-4-(1- ((1-(4- (phenylsulfony...)
Affinity DataIC50: 9nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480097(4-cyclopentyl-2-ethyl-4-(1- ((1-(4-(pyridin-3- yls...)
Affinity DataIC50: 9nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480143(rac-(1S,2R)-2-(4-(1-((1-(4- (cyclopropylsulfonyl)p...)
Affinity DataIC50: 9nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480151(rac-(1S,2R)-2- (cyano(phenyl)(1-((1-(4- (pyridin-4...)
Affinity DataIC50: 9nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480164(rac-(1S,2R)-2- (cyano(phenyl)(1-((1-(4- (phenylsul...)
Affinity DataIC50: 9nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

TargetMenin(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM480179(rac-(1S,2R)-2-(cyano(1-((1- (4-((1-methyl-1H-pyraz...)
Affinity DataIC50: 9nMAssay Description:A fluorescence polarization (FP) competitive binding assay was used to determine the binding affinities of representative menin inhibitors. A FAM lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent

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