Compile Data Set for Download or QSAR
Report error Found 185 Enz. Inhib. hit(s) with all data for entry = 8911
LigandPNGBDBM428786(US10544147, Compound 3-19 | US10544147, Compound 3...)
Affinity DataIC50: 0.700nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
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Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428774((R or S)-1'- (cyclopropanecarbonyl)-5-(9- methyl-8...)
Affinity DataIC50: 1nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
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Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428768(US10544147, Compound 3-2 | (R or S)-1''- (cyclopro...)
Affinity DataIC50: 1nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428749(US10544147, Compound 2-66 | (R or S)-5-(9-ethyl-8-...)
Affinity DataIC50: 1nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
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Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428785(US10544147, Compound 3-18 | (R or S)-1'- (cyclopro...)
Affinity DataIC50: 1.90nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428713(US10544147, Compound 2-30 | (R or S)-3- (cyclobuty...)
Affinity DataIC50: 2nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
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Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428659(US10544147, Compound 1-16 | (R or S)-3-benzyl-5-(9...)
Affinity DataIC50: 2nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428743(US10544147, Compound 2-59 | US10544147, Compound 2...)
Affinity DataIC50: 2nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
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Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428751(US10544147, Compound 2-67 | (R or S)-3-((2-fluoro-...)
Affinity DataIC50: 2nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
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Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428770(US10544147, Compound 3-4 | (R or S)-1''- (cyclopro...)
Affinity DataIC50: 2nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428685(US10544147, Compound 2-2 | (R or S)-5-[9-ethyl-8-(...)
Affinity DataIC50: 2nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
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Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428780((R or S)-1''-isopropyl-5-(9- methyl-8-(2- methylpy...)
Affinity DataIC50: 2nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428783(US10544147, Compound 3-16 | (R or S)-1'- (cyclopro...)
Affinity DataIC50: 2nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428784(US10544147, Compound 3-17 | (R or S)-1'- (cyclopro...)
Affinity DataIC50: 2.5nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428777(US10544147, Compound 3-10 | (R or S)-1'- (cyclopro...)
Affinity DataIC50: 3nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
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Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428679((R or S)-5-(9-ethyl-8-(2- methylpyrimidin-5-yl)-9H...)
Affinity DataIC50: 3nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428778(US10544147, Compound 3-12 | (R or S)-5-(9-ethyl-8-...)
Affinity DataIC50: 3nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428826(US10544147, Compound 5-7 | (R or S)-1-(1- cyclopro...)
Affinity DataIC50: 3nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428739(US10544147, Compound 2-55 | (R or S)-5-(9-ethyl-8-...)
Affinity DataIC50: 3nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428755(US10544147, Compound 2-72 | (R or S)-5-(9-ethyl-8-...)
Affinity DataIC50: 3nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
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Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428673([(R,R) or (R,S) or (S,S) or (S,R)]-5-(9-ethyl-8-(2...)
Affinity DataIC50: 3nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428723((R or S)-3-((5-(9-ethyl-8-(2- methylpyrimidin-5-yl...)
Affinity DataIC50: 3nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428819(US10544147, Compound 4-16 | 6-(9-ethyl-8-(2- methy...)
Affinity DataIC50: 3nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428689(US10544147, Compound 2-6 | (R or S)-1-{5-[9-ethyl-...)
Affinity DataIC50: 3nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428733(US10544147, Compound 2-49 | US10544147, Compound 2...)
Affinity DataIC50: 3nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428663(US10544147, Compound 1-20 | US10544147, Compound 1...)
Affinity DataIC50: 4nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428731(US10544147, Compound 2-47 | (R or S)-5-(9-ethyl-8-...)
Affinity DataIC50: 4nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428788(US10544147, Compound 3-21 | (R or S)-5-(9-ethyl-8-...)
Affinity DataIC50: 4nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428644(US10544147, Compound 1-1 | US10544147, Compound 1-...)
Affinity DataIC50: 4nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428806(US10544147, Compound 4-3 | (R or S)-6-[9-ethyl-8-(...)
Affinity DataIC50: 4nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428737(US10544147, Compound 2-53 | US10544147, Compound 2...)
Affinity DataIC50: 4nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428719(US10544147, Compound 2-36 | 5-[9-ethyl-8-(2- methy...)
Affinity DataIC50: 4nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428753(US10544147, Compound 2-69 | (R or S)-3-((2,2- difl...)
Affinity DataIC50: 4nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428668((R or S)-3- (cyclopropylmethyl)-5-(9- ethyl-8-(1-e...)
Affinity DataIC50: 4nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428824(US10544147, Compound 5-5 | (R or S)-3-(1- cyclopro...)
Affinity DataIC50: 5nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428696(US10544147, Compound 2-13 | 3-{[(1S)-1- cyclopropy...)
Affinity DataIC50: 5nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428776(US10544147, Compound 3-9 | (R or S)-1'- (cycloprop...)
Affinity DataIC50: 5nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428725(US10544147, Compound 2-42 | (R or S)-3-((2,2- difl...)
Affinity DataIC50: 5nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428727(US10544147, Compound 2-43 | (R or S)-5-(9-ethyl-8-...)
Affinity DataIC50: 5nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428677(US10544147, Compound 1-35 | (R or S)-5-(9-ethyl-8-...)
Affinity DataIC50: 5nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428687(US10544147, Compound 2-4 | (R or S)-3-[(cis)-2,6- ...)
Affinity DataIC50: 5nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428813(US10544147, Compound 4-11 | (R or S)-3-benzyl-5-[9...)
Affinity DataIC50: 5nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428669((R or S)-3-isobutyl-3-methyl- 5-(9-methyl-8-(2- me...)
Affinity DataIC50: 5nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428782(US10544147, Compound 3-15 | (R or S)-1'- (cyclopro...)
Affinity DataIC50: 5nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428808(US10544147, Compound 4-5 | (R or S)-9-ethyl-6-[3- ...)
Affinity DataIC50: 6nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428745(US10544147, Compound 2-62 | 3-(R or S)-((3R,4R)-3,...)
Affinity DataIC50: 6nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428790((R or S)-5-(9-ethyl-8-(2- methylpyrimidin-5-yl)-9H...)
Affinity DataIC50: 6nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428747((R or S)-5-(9-ethyl-8-(2- methylpyrimidin-5-yl)-9H...)
Affinity DataIC50: 6nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428735(US10544147, Compound 2-51 | US10544147, Compound 2...)
Affinity DataIC50: 6nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
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Date in BDB:
11/2/2020
Entry Details
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LigandPNGBDBM428729(US10544147, Compound 2-45 | US10544147, Compound 2...)
Affinity DataIC50: 7nMAssay Description:The PI3-Kinase biochemical assays were developed to measure the intrinsic potency and compound dependent inhibition of the alpha, beta, delta, and ga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2020
Entry Details
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