Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 1153
TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM310976(US10155733, Strucure 3e | US10155733, Example 5)
Affinity DataIC50: 9.5nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2019
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TargetMuscarinic acetylcholine receptor M3(Human)
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LigandPNGBDBM311052(US10155733, Strucure 3g | US10155733, Example 7)
Affinity DataIC50: 60nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2019
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TargetMuscarinic acetylcholine receptor M3(Human)
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LigandPNGBDBM311058(US10155733, Strucure 7d | US10155733, Example 11)
Affinity DataIC50: 63nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2019
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TargetMuscarinic acetylcholine receptor M3(Human)
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LigandPNGBDBM311061(US10155733, Strucure 7g | US10155733, Example 14)
Affinity DataIC50: 144nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2019
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TargetMuscarinic acetylcholine receptor M3(Human)
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LigandPNGBDBM311059(US10155733, Strucure 7e | US10155733, Example 12)
Affinity DataIC50: 195nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2019
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM311064(US10155733, Strucure 7j | US10155733, Example 17)
Affinity DataIC50: 266nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
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TargetMuscarinic acetylcholine receptor M3(Human)
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LigandPNGBDBM311070(US10155733, Strucure 9f | US10155733, Example 23)
Affinity DataIC50: 346nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2019
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TargetMuscarinic acetylcholine receptor M3(Human)
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LigandPNGBDBM311068(US10155733, Strucure 9d | US10155733, Example 21)
Affinity DataIC50: 357nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM311051(US10155733, Strucure 3f | US10155733, Example 6)
Affinity DataIC50: 409nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2019
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM311056(US10155733, Strucure 7c | US10155733, Example 10)
Affinity DataIC50: 599nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
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LigandPNGBDBM311066(US10155733, Strucure 9b | US10155733, Example 19)
Affinity DataIC50: 609nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2019
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM311067(US10155733, Strucure 9c | US10155733, Example 20)
Affinity DataIC50: 1.20E+3nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM311074(US10155733, Strucure 13 | US10155733, Example 27)
Affinity DataIC50: 1.40E+3nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM310964(US10155733, Strucure 3c | US10155733, Example 3)
Affinity DataIC50: 1.40E+3nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM311053(US10155733, Strucure 7a | US10155733, Example 8)
Affinity DataIC50: 1.80E+3nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM311054(US10155733, Strucure 7b | US10155733, Example 9)
Affinity DataIC50: 2.10E+3nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
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TargetMuscarinic acetylcholine receptor M3(Human)
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LigandPNGBDBM310951(US10155733, Strucure 3b | US10155733, Example 2)
Affinity DataIC50: 2.10E+3nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM311072(US10155733, Strucure 9h | US10155733, Example 25)
Affinity DataIC50: 2.70E+3nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM311062(US10155733, Strucure 7h | US10155733, Example 15)
Affinity DataIC50: 3.00E+3nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM311071(US10155733, Strucure 9g | US10155733, Example 24)
Affinity DataIC50: 3.90E+3nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM311073(US10155733, Strucure 11 | US10155733, Example 26)
Affinity DataIC50: 4.30E+3nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM311063(US10155733, Strucure 7i | US10155733, Example 16)
Affinity DataIC50: 4.60E+3nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM311060(US10155733, Strucure 7f | US10155733, Example 13)
Affinity DataIC50: 4.70E+3nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM310949(US10155733, Strucure 3a | US10155733, Example 1)
Affinity DataIC50: 5.30E+3nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM311069(US10155733, Strucure 9e | US10155733, Example 22)
Affinity DataIC50: 5.70E+3nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM311065(US10155733, Strucure 9a | US10155733, Example 18)
Affinity DataIC50: 6.00E+3nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
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TargetMuscarinic acetylcholine receptor M3(Human)
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US Patent
LigandPNGBDBM310972(US10155733, Strucure 3d | US10155733, Example 4)
Affinity DataIC50: 7.90E+3nMAssay Description:The muscarinic 3 receptor binding assay was adapted from Perkin Elmer. Briefly, assay buffer (60 μL of pH 7.4 phosphate saline buffer) was added...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
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