Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 5030
TargetSubstance-P receptor(Human)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Guinea pig)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Human)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50071112(SR 48968 | CHEMBL56835 | N-[4-(4-Acetylamino-4-phe...)
Affinity DataKi:  0.440nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Guinea pig)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50000040(CHEMBL16192 | (+)(2-Benzhydryl-1-aza-bicyclo[2.2.2...)
Affinity DataKi:  0.550nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Human)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM81942(Neurokinin alpha | NSC_55582 | NKA | CAS_55582 | S...)
Affinity DataKi:  0.650nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Bovine)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50071112(SR 48968 | CHEMBL56835 | N-[4-(4-Acetylamino-4-phe...)
Affinity DataKi:  0.710nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Bovine)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM81942(Neurokinin alpha | NSC_55582 | NKA | CAS_55582 | S...)
Affinity DataKi:  0.960nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Rat)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataKi:  1.02nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Human)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50030178(FK 888 | CHEMBL303548 | (R)-4-Hydroxy-1-(1-methyl-...)
Affinity DataKi:  1.49nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Golden hamster)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM81942(Neurokinin alpha | NSC_55582 | NKA | CAS_55582 | S...)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Guinea pig)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175522(CHEMBL372587 | MDL 105,212 (R)-enantiomer | 1-{2-[...)
Affinity DataKi:  2.12nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Guinea pig)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM84953(MDL 105,212A (R)-enantiomer)
Affinity DataKi:  2.99nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Human)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175522(CHEMBL372587 | MDL 105,212 (R)-enantiomer | 1-{2-[...)
Affinity DataKi:  3.11nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Guinea pig)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50030178(FK 888 | CHEMBL303548 | (R)-4-Hydroxy-1-(1-methyl-...)
Affinity DataKi:  3.13nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetNeuromedin-K receptor(Guinea pig)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM81944(NSC_5311312 | NKB | CAS_86933-75-7 | neuromedin K)
Affinity DataKi:  3.54nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Human)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM84953(MDL 105,212A (R)-enantiomer)
Affinity DataKi:  3.69nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Guinea pig)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50290297(CHEMBL539021 | MDL 103,392A racemate | 1-{2-[(R)-3...)
Affinity DataKi:  5.88nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Golden hamster)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175522(CHEMBL372587 | MDL 105,212 (R)-enantiomer | 1-{2-[...)
Affinity DataKi:  6.98nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Human)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50290297(CHEMBL539021 | MDL 103,392A racemate | 1-{2-[(R)-3...)
Affinity DataKi:  7.07nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Golden hamster)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50071112(SR 48968 | CHEMBL56835 | N-[4-(4-Acetylamino-4-phe...)
Affinity DataKi:  7.32nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Human)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM84953(MDL 105,212A (R)-enantiomer)
Affinity DataKi:  7.93nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Rat)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50029885(RP-67580 | RP 67,580 | 2-[1-Imino-2-(2-methoxy-phe...)
Affinity DataKi:  8.29nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Human)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175522(CHEMBL372587 | MDL 105,212 (R)-enantiomer | 1-{2-[...)
Affinity DataKi:  8.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Bovine)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM84953(MDL 105,212A (R)-enantiomer)
Affinity DataKi:  8.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Bovine)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175522(CHEMBL372587 | MDL 105,212 (R)-enantiomer | 1-{2-[...)
Affinity DataKi:  8.49nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Rat)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50000040(CHEMBL16192 | (+)(2-Benzhydryl-1-aza-bicyclo[2.2.2...)
Affinity DataKi:  15.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetNeuromedin-K receptor(Guinea pig)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175522(CHEMBL372587 | MDL 105,212 (R)-enantiomer | 1-{2-[...)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Human)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50290297(CHEMBL539021 | MDL 103,392A racemate | 1-{2-[(R)-3...)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Guinea pig)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50029885(RP-67580 | RP 67,580 | 2-[1-Imino-2-(2-methoxy-phe...)
Affinity DataKi:  36nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetNeuromedin-K receptor(Guinea pig)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50290297(CHEMBL539021 | MDL 103,392A racemate | 1-{2-[(R)-3...)
Affinity DataKi:  54.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Guinea pig)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM84954(CAS_6437864 | NSC_6437864 | FK 224)
Affinity DataKi:  98.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Human)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175494(1-{2-[(R)-3-(3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  160nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Guinea pig)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175494(1-{2-[(R)-3-(3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  183nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Bovine)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175494(1-{2-[(R)-3-(3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  207nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetNeuromedin-K receptor(Guinea pig)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50071112(SR 48968 | CHEMBL56835 | N-[4-(4-Acetylamino-4-phe...)
Affinity DataKi:  208nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Human)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM84954(CAS_6437864 | NSC_6437864 | FK 224)
Affinity DataKi:  215nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Guinea pig)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50071112(SR 48968 | CHEMBL56835 | N-[4-(4-Acetylamino-4-phe...)
Affinity DataKi:  217nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Rat)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM84954(CAS_6437864 | NSC_6437864 | FK 224)
Affinity DataKi:  228nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Bovine)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM84954(CAS_6437864 | NSC_6437864 | FK 224)
Affinity DataKi:  311nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Rat)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175522(CHEMBL372587 | MDL 105,212 (R)-enantiomer | 1-{2-[...)
Affinity DataKi:  408nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Human)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM84954(CAS_6437864 | NSC_6437864 | FK 224)
Affinity DataKi:  434nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Human)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50071112(SR 48968 | CHEMBL56835 | N-[4-(4-Acetylamino-4-phe...)
Affinity DataKi:  593nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Golden hamster)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175494(1-{2-[(R)-3-(3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  711nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Human)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175494(1-{2-[(R)-3-(3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  760nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Human)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50030178(FK 888 | CHEMBL303548 | (R)-4-Hydroxy-1-(1-methyl-...)
Affinity DataKi:  1.52E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Rat)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50030178(FK 888 | CHEMBL303548 | (R)-4-Hydroxy-1-(1-methyl-...)
Affinity DataKi:  2.07E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-P receptor(Rat)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175494(1-{2-[(R)-3-(3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  2.20E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetNeuromedin-K receptor(Guinea pig)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM50175494(1-{2-[(R)-3-(3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  2.31E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetNeuromedin-K receptor(Guinea pig)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM84954(CAS_6437864 | NSC_6437864 | FK 224)
Affinity DataKi:  3.56E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
TargetSubstance-K receptor(Golden hamster)
Hoechst Marion Roussel

Curated by PDSP Ki Database
LigandPNGBDBM84954(CAS_6437864 | NSC_6437864 | FK 224)
Affinity DataKi:  3.59E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details
PubMed
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