Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50029660
TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286614(Sodium; 2-[2-{2-[(2,6-dimethyl-piperidine-1-carbon...)
Affinity DataIC50: 1.20nMAssay Description:Antagonistic activity against endothelin B (ETB) receptor using human girardi heart cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286622(Ac-W-F-F-N-Y-Y-W | CHEMBL405677)
Affinity DataIC50: 250nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286614(Sodium; 2-[2-{2-[(2,6-dimethyl-piperidine-1-carbon...)
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonistic activity against endothelin A (ETA) receptor using human neuroblastoma cell line.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286619(Ac-bhg-F-N-Y-Y-W | CHEMBL385405)
Affinity DataIC50: 1.90E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286618(W-F-F-N--Y-Y-W | CHEMBL413880)
Affinity DataIC50: 2.40E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286620(W-H-G-T-A-P-D-W-F-F-N-Y-Y-W | CHEMBL415614)
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286616(G-N-W-H-G-T-A-P-D-W-F-F-N-Y-Y-W | CHEMBL267610)
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286616(G-N-W-H-G-T-A-P-D-W-F-F-N-Y-Y-W | CHEMBL267610)
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286620(W-H-G-T-A-P-D-W-F-F-N-Y-Y-W | CHEMBL415614)
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286619(Ac-bhg-F-N-Y-Y-W | CHEMBL385405)
Affinity DataIC50: 4.30E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286613(Cyclic (Gly1-Asp9) (Gly-Asn-Trp-His-Gly-Thr-Ala-Pr...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286613(Cyclic (Gly1-Asp9) (Gly-Asn-Trp-His-Gly-Thr-Ala-Pr...)
Affinity DataIC50: 6.50E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286613(Cyclic (Gly1-Asp9) (Gly-Asn-Trp-His-Gly-Thr-Ala-Pr...)
Affinity DataIC50: 6.50E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286622(Ac-W-F-F-N-Y-Y-W | CHEMBL405677)
Affinity DataIC50: 7.60E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286613(Cyclic (Gly1-Asp9) (Gly-Asn-Trp-His-Gly-Thr-Ala-Pr...)
Affinity DataIC50: 7.60E+3nMAssay Description:Ability to block endothelin-1 (ET-1) stimulated arachidonic acid release in rabbit renal vascular smooth muscle cells (AARA) expressing recombinant r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286613(Cyclic (Gly1-Asp9) (Gly-Asn-Trp-His-Gly-Thr-Ala-Pr...)
Affinity DataIC50: 7.80E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286615(Ac-w-F-F-N-Y-Y-W | CHEMBL441006)
Affinity DataIC50: 8.10E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286617(bhg-F-N-Y-Y-W | CHEMBL414917)
Affinity DataIC50: 9.50E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286617(bhg-F-N-Y-Y-W | CHEMBL414917)
Affinity DataIC50: 1.30E+4nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286615(Ac-w-F-F-N-Y-Y-W | CHEMBL441006)
Affinity DataIC50: 1.40E+4nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286618(W-F-F-N--Y-Y-W | CHEMBL413880)
Affinity DataIC50: 1.50E+4nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286613(Cyclic (Gly1-Asp9) (Gly-Asn-Trp-His-Gly-Thr-Ala-Pr...)
Affinity DataIC50: 1.60E+4nMAssay Description:Ability to block sarafotoxin-6c (SRTX-6c) stimulated arachidonic acid release in chinese hamster ovary (CHO) cells expressing recombinant rat endothe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin receptor type B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286621(F-F-N-Y-YW | CHEMBL264253)
Affinity DataIC50: 2.50E+4nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286621(F-F-N-Y-YW | CHEMBL264253)
Affinity DataIC50: 2.50E+4nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article