Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50019007
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50118359((2-Chloro-7,7-dioxo-4,7-dihydro-1,7-dithia-4,6-dia...)
Affinity DataEC50:  750nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614565(CHEMBL5291159)
Affinity DataEC50:  550nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614566(CHEMBL5279052)
Affinity DataEC50:  970nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614567(CHEMBL5280335)
Affinity DataEC50:  940nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614568(CHEMBL5270996)
Affinity DataEC50:  560nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614569(CHEMBL5268632)
Affinity DataEC50:  1.10E+3nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614570(CHEMBL5267062)
Affinity DataEC50:  310nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614571(CHEMBL5270814)
Affinity DataEC50:  570nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614572(CHEMBL5270566)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614564(CHEMBL5285592)
Affinity DataEC50:  880nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614573(CHEMBL5284807)
Affinity DataEC50:  7.00E+3nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50237612(CHEBI:4495 | Diazoxide | Eudemine | Eudimine | Hyp...)
Affinity DataEC50:  3.00E+4nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614574(CHEMBL5274079)
Affinity DataEC50:  2.51E+3nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614575(CHEMBL5275196)
Affinity DataEC50:  3.73E+3nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614576(CHEMBL5290652)
Affinity DataEC50:  7.42E+3nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614577(CHEMBL5285443)
Affinity DataEC50:  100nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50118359((2-Chloro-7,7-dioxo-4,7-dihydro-1,7-dithia-4,6-dia...)
Affinity DataEC50:  450nMAssay Description:Activation of human Kir6.2/SUR1 channel outward current expressed in HEK293 cells at -70 mV holding potential by EPC9 patch-clamp amplifier based ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50409914(BMS-191095)
Affinity DataEC50:  1.40E+3nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel openingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614555(CHEMBL5283293)
Affinity DataEC50:  2.00E+3nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614547(CHEMBL5273292)
Affinity DataEC50:  460nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614548(CHEMBL5273275)
Affinity DataEC50:  250nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614549(CHEMBL5286136)
Affinity DataEC50:  660nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614550(CHEMBL5283421)
Affinity DataEC50:  780nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614551(CHEMBL5277742)
Affinity DataEC50:  1.10E+3nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614552(CHEMBL5266806)
Affinity DataEC50:  1.00E+3nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614553(CHEMBL5285581)
Affinity DataEC50:  3.30E+3nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614554(CHEMBL5273158)
Affinity DataEC50:  3.50E+4nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614546(CHEMBL5276858)
Affinity DataEC50:  1.80E+3nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614556(CHEMBL5273874)
Affinity DataEC50:  6.50E+3nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614557(CHEMBL5288579)
Affinity DataEC50:  4.10E+3nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614558(CHEMBL5288853)
Affinity DataEC50:  1.14E+3nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614559(CHEMBL5291259)
Affinity DataEC50:  530nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614560(CHEMBL5280182)
Affinity DataEC50:  710nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614561(CHEMBL5269505)
Affinity DataEC50:  710nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614562(CHEMBL5276527)
Affinity DataEC50:  1.00E+3nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50614563(CHEMBL5286203)
Affinity DataEC50:  3.10E+3nMAssay Description:Activation of Kir6.2/SUR1 (unknown origin) channel opening expressed in human T-REx-293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed