Compile Data Set for Download or QSAR
Report error Found 71 Enz. Inhib. hit(s) with all data for entry = 50015522
TargetBromodomain-containing protein 7(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587251(CHEMBL5080049)
Affinity DataKd:  230nMAssay Description:Binding affinity to human BRD7 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587255(CHEMBL5080169)
Affinity DataKd:  8.26E+3nMAssay Description:Binding affinity to human BRD4 domain 1 (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587250(CHEMBL5077168)
Affinity DataKd:  2.98E+3nMAssay Description:Binding affinity to human BRD4 domain 1 (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587256(CHEMBL5079915)
Affinity DataKd:  2.66E+3nMAssay Description:Binding affinity to human BRD4 domain 1 (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587257(CHEMBL5092849)
Affinity DataKd:  3.67E+3nMAssay Description:Binding affinity to human BRD4 domain 1 (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587251(CHEMBL5080049)
Affinity DataKd:  790nMAssay Description:Binding affinity to human BRD4 domain 1 (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587252(CHEMBL5083849)
Affinity DataKd:  76nMAssay Description:Binding affinity to human BRD4 domain 1 (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587258(CHEMBL5091031)
Affinity DataKd:  34nMAssay Description:Binding affinity to human BRD4 domain 1 (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 7(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587252(CHEMBL5083849)
Affinity DataKd:  125nMAssay Description:Binding affinity to human BRD7 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50158909(CHEMBL3787231)
Affinity DataKd:  160nMAssay Description:Binding affinity to human BRD4 domain 1 (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 7(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587250(CHEMBL5077168)
Affinity DataKd:  8.50E+3nMAssay Description:Binding affinity to human BRD7 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 7(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587249(CHEMBL5094795)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human BRD7 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587252(CHEMBL5083849)
Affinity DataKd:  100nMAssay Description:Binding affinity to human BRD3 domain 2 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587251(CHEMBL5080049)
Affinity DataKd:  3.75E+3nMAssay Description:Binding affinity to human BRD3 domain 2 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587250(CHEMBL5077168)
Affinity DataKd:  7.55E+3nMAssay Description:Binding affinity to human BRD3 domain 2 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587249(CHEMBL5094795)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human BRD3 domain 1 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50158909(CHEMBL3787231)
Affinity DataKd:  490nMAssay Description:Binding affinity to human BRD3 domain 2 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587249(CHEMBL5094795)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human BRD3 domain 2 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587252(CHEMBL5083849)
Affinity DataKd:  67nMAssay Description:Binding affinity to human BRD2 domain 2 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50158909(CHEMBL3787231)
Affinity DataKd:  380nMAssay Description:Binding affinity to human BRD3 domain 1 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587250(CHEMBL5077168)
Affinity DataKd:  5.65E+3nMAssay Description:Binding affinity to human BRD3 domain 1 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587251(CHEMBL5080049)
Affinity DataKd:  1.50E+3nMAssay Description:Binding affinity to human BRD3 domain 1 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587252(CHEMBL5083849)
Affinity DataKd:  37nMAssay Description:Binding affinity to human BRD3 domain 1 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587249(CHEMBL5094795)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human BRD2 domain 2 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50158909(CHEMBL3787231)
Affinity DataKd:  830nMAssay Description:Binding affinity to human BRD2 domain 2 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587250(CHEMBL5077168)
Affinity DataKd:  3.30E+3nMAssay Description:Binding affinity to human BRD2 domain 2 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587251(CHEMBL5080049)
Affinity DataKd:  3.10E+3nMAssay Description:Binding affinity to human BRD2 domain 2 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587254(CHEMBL5069833)
Affinity DataKd:  6.92E+3nMAssay Description:Binding affinity to human BRD4 domain 1 (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587249(CHEMBL5094795)
Affinity DataKd:  7.70E+3nMAssay Description:Binding affinity to human BRD2 domain 1 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50158909(CHEMBL3787231)
Affinity DataKd:  170nMAssay Description:Binding affinity to human BRD2 domain 1 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587250(CHEMBL5077168)
Affinity DataKd:  7.40E+3nMAssay Description:Binding affinity to human BRD2 domain 1 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587251(CHEMBL5080049)
Affinity DataKd:  230nMAssay Description:Binding affinity to human BRD2 domain 1 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587252(CHEMBL5083849)
Affinity DataKd:  27nMAssay Description:Binding affinity to human BRD2 domain 1 assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587253(CHEMBL5094765)
Affinity DataKd:  1.15E+4nMAssay Description:Binding affinity to human BRD4 domain 1 (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587249(CHEMBL5094795)
Affinity DataKd:  4.50E+3nMAssay Description:Binding affinity to human BRD4 domain 1 (unknown origin) assessed as dissociation constant by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587250(CHEMBL5077168)
Affinity DataIC50: 42nMAssay Description:Inhibition of human recombinant HDAC6 assessed as fluorescence using fluorogenic substrate ZMAL incubated for 90 min by microplate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587249(CHEMBL5094795)
Affinity DataIC50: 45nMAssay Description:Inhibition of human recombinant HDAC6 assessed as fluorescence using fluorogenic substrate ZMAL incubated for 90 min by microplate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587251(CHEMBL5080049)
Affinity DataIC50: 46nMAssay Description:Inhibition of human recombinant HDAC6 assessed as fluorescence using fluorogenic substrate ZMAL incubated for 90 min by microplate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 51nMAssay Description:Inhibition of human recombinant HDAC6 assessed as fluorescence using fluorogenic substrate ZMAL incubated for 90 min by microplate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587251(CHEMBL5080049)
Affinity DataIC50: 64nMAssay Description:Inhibition of human HDAC3 assessed as target activity using fluorogenic substrate ZMAL for 90 min by microplate reader at 355nmMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587252(CHEMBL5083849)
Affinity DataIC50: 67nMAssay Description:Inhibition of human recombinant HDAC6 assessed as fluorescence using fluorogenic substrate ZMAL incubated for 90 min by microplate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587257(CHEMBL5092849)
Affinity DataIC50: 73nMAssay Description:Inhibition of human recombinant HDAC6 assessed as fluorescence using fluorogenic substrate ZMAL incubated for 90 min by microplate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587256(CHEMBL5079915)
Affinity DataIC50: 80nMAssay Description:Inhibition of human recombinant HDAC6 assessed as fluorescence using fluorogenic substrate ZMAL incubated for 90 min by microplate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587251(CHEMBL5080049)
Affinity DataIC50: 93nMAssay Description:Inhibition of human recombinant HDAC1 assessed as fluorescence using fluorogenic substrate ZMAL incubated for 90 min by microplate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587257(CHEMBL5092849)
Affinity DataIC50: 97nMAssay Description:Inhibition of human recombinant HDAC1 assessed as fluorescence using fluorogenic substrate ZMAL incubated for 90 min by microplate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 108nMAssay Description:Inhibition of human HDAC3 assessed as target activity using fluorogenic substrate ZMAL for 90 min by microplate reader at 355nmMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587250(CHEMBL5077168)
Affinity DataIC50: 119nMAssay Description:Inhibition of human HDAC3 assessed as target activity using fluorogenic substrate ZMAL for 90 min by microplate reader at 355nmMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 120nMAssay Description:Inhibition of human recombinant HDAC1 assessed as fluorescence using fluorogenic substrate ZMAL incubated for 90 min by microplate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 1(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587249(CHEMBL5094795)
Affinity DataIC50: 125nMAssay Description:Inhibition of human recombinant HDAC1 assessed as fluorescence using fluorogenic substrate ZMAL incubated for 90 min by microplate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Universit£T Leipzig

Curated by ChEMBL
LigandPNGBDBM50587256(CHEMBL5079915)
Affinity DataIC50: 142nMAssay Description:Inhibition of human recombinant HDAC1 assessed as fluorescence using fluorogenic substrate ZMAL incubated for 90 min by microplate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
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