Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 50014020
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 1nMAssay Description:Inhibition of APN (unknown origin) using Ala-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571866(CHEMBL4862557)
Affinity DataIC50: 34nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 52nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571865(CHEMBL4863142)
Affinity DataIC50: 99nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571867(CHEMBL4875461)
Affinity DataIC50: 115nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571872(CHEMBL4864508)
Affinity DataIC50: 120nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571874(CHEMBL4855038)
Affinity DataIC50: 151nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571868(CHEMBL4854530)
Affinity DataIC50: 262nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571862(CHEMBL4847534)
Affinity DataIC50: 275nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571856(CHEMBL4850551)
Affinity DataIC50: 377nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571857(CHEMBL4854083)
Affinity DataIC50: 698nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571871(CHEMBL4873254)
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571864(CHEMBL4853997)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571858(CHEMBL4855147)
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571869(CHEMBL4852033)
Affinity DataIC50: 1.76E+3nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571873(CHEMBL4877678)
Affinity DataIC50: 1.76E+3nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571870(CHEMBL4849207)
Affinity DataIC50: 1.97E+3nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571859(CHEMBL4863578)
Affinity DataIC50: 2.68E+3nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571863(CHEMBL4846862)
Affinity DataIC50: 4.44E+3nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571860(CHEMBL4858634)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571861(CHEMBL4873293)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571856(CHEMBL4850551)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of APN (unknown origin) using Ala-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571857(CHEMBL4854083)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of APN (unknown origin) using Ala-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571864(CHEMBL4853997)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of ERAP2 (unknown origin) using Arg-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571864(CHEMBL4853997)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of APN (unknown origin) using Ala-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571865(CHEMBL4863142)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of APN (unknown origin) using Ala-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571874(CHEMBL4855038)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of ERAP2 (unknown origin) using Arg-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571866(CHEMBL4862557)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of APN (unknown origin) using Ala-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571867(CHEMBL4875461)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of APN (unknown origin) using Ala-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571868(CHEMBL4854530)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of APN (unknown origin) using Ala-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571869(CHEMBL4852033)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of APN (unknown origin) using Ala-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571871(CHEMBL4873254)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of APN (unknown origin) using Ala-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571872(CHEMBL4864508)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of APN (unknown origin) using Ala-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571873(CHEMBL4877678)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of APN (unknown origin) using Ala-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571874(CHEMBL4855038)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of APN (unknown origin) using Ala-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571872(CHEMBL4864508)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of ERAP2 (unknown origin) using Arg-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571856(CHEMBL4850551)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin) using midazolam as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571857(CHEMBL4854083)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin) using midazolam as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571856(CHEMBL4850551)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin) using testosterone as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571857(CHEMBL4854083)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin) using testosterone as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571856(CHEMBL4850551)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of ERAP2 (unknown origin) using Arg-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571857(CHEMBL4854083)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of ERAP2 (unknown origin) using Arg-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571865(CHEMBL4863142)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of ERAP2 (unknown origin) using Arg-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571866(CHEMBL4862557)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of ERAP2 (unknown origin) using Arg-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571867(CHEMBL4875461)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of ERAP2 (unknown origin) using Arg-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571868(CHEMBL4854530)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of ERAP2 (unknown origin) using Arg-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571869(CHEMBL4852033)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of ERAP2 (unknown origin) using Arg-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571871(CHEMBL4873254)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of ERAP2 (unknown origin) using Arg-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 2(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571873(CHEMBL4877678)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of ERAP2 (unknown origin) using Arg-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50571877(CHEMBL4878272)
Affinity DataKi:  1.51E+5nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
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