Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50011433
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50546904(CHEMBL4743669)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50300690(CHEMBL576982 | N-(5-tert-Butyl-isoxazol-3-yl)-N'-{...)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50546908(CHEMBL4749162)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50546906(CHEMBL4757873)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50546903(CHEMBL4763985)
Affinity DataIC50: 21nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50546907(CHEMBL4740352)
Affinity DataIC50: 83nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50546909(CHEMBL4795939)
Affinity DataIC50: 109nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50546905(CHEMBL4754456)
Affinity DataIC50: 157nMAssay Description:Inhibition of FLT3 ITD mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed