Compile Data Set for Download or QSAR
Report error Found 111 Enz. Inhib. hit(s) with all data for entry = 50010368
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 221048BDBM221048(US9303017, Varenicline | US9284322, varenicline)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538045BDBM50538045(CHEMBL4636163)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538008BDBM50538008(CHEMBL4638732)
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538047BDBM50538047(CHEMBL4647019)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538046BDBM50538046(CHEMBL4647198)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538027BDBM50538027(CHEMBL4644169)
Affinity DataKi:  0.370nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538033BDBM50538033(CHEMBL4648557)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538030BDBM50538030(CHEMBL4638919)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538038BDBM50538038(CHEMBL4648098)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538036BDBM50538036(CHEMBL4634253)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538063BDBM50538063(CHEMBL4642118)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82070BDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538014BDBM50538014(CHEMBL4637076)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538035BDBM50538035(CHEMBL4634110)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538029BDBM50538029(CHEMBL4648968)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538041BDBM50538041(CHEMBL4642769)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538064BDBM50538064(CHEMBL4642865)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538028BDBM50538028(CHEMBL4634727)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538039BDBM50538039(CHEMBL4637371)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538022BDBM50538022(CHEMBL4649539)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538037BDBM50538037(CHEMBL4645367)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538062BDBM50538062(CHEMBL4637698)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538057BDBM50538057(CHEMBL4643942)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538046BDBM50538046(CHEMBL4647198)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in IMR32 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538051BDBM50538051(CHEMBL4641432)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538061BDBM50538061(CHEMBL4640279)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538060BDBM50538060(CHEMBL4645127)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257941BDBM50257941(7-(pyridin-3-yl)-1,7-diazaspiro[4.4]nonane | CHEMB...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538024BDBM50538024(CHEMBL4646061)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538054BDBM50538054(CHEMBL4642287)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538045BDBM50538045(CHEMBL4636163)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in IMR32 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538059BDBM50538059(CHEMBL4639792)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50056147BDBM50056147(ABT-089 | 2-Methyl-3-((S)-1-pyrrolidin-2-ylmethoxy...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538025BDBM50538025(CHEMBL4634566)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538053BDBM50538053(CHEMBL4646023)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538026BDBM50538026(CHEMBL4640410)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538021BDBM50538021(CHEMBL4641810)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 221048BDBM221048(US9303017, Varenicline | US9284322, varenicline)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in IMR32 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538066BDBM50538066(CHEMBL4640566)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538051BDBM50538051(CHEMBL4641432)
Affinity DataKi:  68nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR expressed in IMR32 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538011BDBM50538011(CHEMBL4636272)
Affinity DataKi:  131nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538009BDBM50538009(CHEMBL4646643)
Affinity DataKi:  149nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538023BDBM50538023(CHEMBL4637361)
Affinity DataKi:  231nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538048BDBM50538048(CHEMBL4642328)
Affinity DataKi:  242nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538010BDBM50538010(CHEMBL4637625)
Affinity DataKi:  265nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538034BDBM50538034(CHEMBL4638726)
Affinity DataKi:  327nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538056BDBM50538056(CHEMBL4634584)
Affinity DataKi:  327nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538040BDBM50538040(CHEMBL4649507)
Affinity DataKi:  329nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538050BDBM50538050(CHEMBL4640672)
Affinity DataKi:  341nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538055BDBM50538055(CHEMBL4636268)
Affinity DataKi:  395nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
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