Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50010363
TargetTyrosine-protein kinase JAK1(Human)
Brigham Young University

Curated by ChEMBL
LigandPNGBDBM50537996(CHEMBL4632827)
Affinity DataKd:  550nMAssay Description:Binding affinity to wild-type human partial length JAK1 JH2 pseudokinase domain (R537 to D855 residues) expressed in mammalian expression system at 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Human)
Brigham Young University

Curated by ChEMBL
LigandPNGBDBM50537996(CHEMBL4632827)
Affinity DataKd:  410nMAssay Description:Binding affinity to wild-type human partial length PIK3C3 (S282 to H879 residues) expressed in mammalian expression system at 10 uM by Kinomescan met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed