Compile Data Set for Download or QSAR
Report error Found 84 Enz. Inhib. hit(s) with all data for entry = 50002357
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457545(CHEMBL4210286)
Affinity DataEC50:  248nMAssay Description:Inverse agonist activity at GAL4 DNA-binding domain-tagged RARabetaa (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457563(CHEMBL4205733)
Affinity DataEC50:  0.920nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50048280(6-(3-adamantan-1-yl-4-methoxyphenyl)naphthalene-2-...)
Affinity DataEC50:  3.10nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457565(CHEMBL3910072)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457560(CHEMBL3939687)
Affinity DataEC50:  14nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457552(CHEMBL4210595)
Affinity DataEC50:  3.80nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457543(CHEMBL3934863)
Affinity DataEC50:  9.5nMAssay Description:Inverse agonist activity at GAL4 DNA-binding domain-tagged RARabetaa (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457546(CHEMBL4206237)
Affinity DataEC50:  5nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457566(CHEMBL4211171)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457553(CHEMBL4210099)
Affinity DataEC50:  26nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457567(CHEMBL3891815)
Affinity DataEC50:  20nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457548(CD-5789 | Trifarotene)
Affinity DataEC50:  7.70nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457543(CHEMBL3934863)
Affinity DataEC50:  53nMAssay Description:Inverse agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457566(CHEMBL4211171)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457548(CD-5789 | Trifarotene)
Affinity DataEC50:  125nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457567(CHEMBL3891815)
Affinity DataEC50:  35nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457561(CHEMBL3916016)
Affinity DataEC50:  60nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457554(CHEMBL4202830)
Affinity DataEC50:  40nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457564(CHEMBL4215021)
Affinity DataEC50:  13nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457563(CHEMBL4205733)
Affinity DataEC50:  6.80nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457551(CHEMBL4217953)
Affinity DataEC50:  40nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457564(CHEMBL4215021)
Affinity DataEC50:  8nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50048291(6-[3'-(1-adamantyl)-4'-hydroxyphenyl]-2-naphthalen...)
Affinity DataEC50:  226nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457550(CHEMBL4207978)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457567(CHEMBL3891815)
Affinity DataEC50:  270nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457554(CHEMBL4202830)
Affinity DataEC50:  317nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457552(CHEMBL4210595)
Affinity DataEC50:  43nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM31888(CD666)
Affinity DataEC50:  370nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457565(CHEMBL3910072)
Affinity DataEC50:  918nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457547(CHEMBL3953756)
Affinity DataEC50:  10nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457570(CHEMBL4207786)
Affinity DataEC50:  15nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457569(CHEMBL4205304)
Affinity DataEC50:  279nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457562(CHEMBL4203742)
Affinity DataEC50:  8.60nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457562(CHEMBL4203742)
Affinity DataEC50:  22nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457542(CHEMBL4212472)
Affinity DataEC50:  11nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM31888(CD666)
Affinity DataEC50:  140nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457568(CHEMBL4211195)
Affinity DataEC50:  168nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM393289(US9963439, BMS961)
Affinity DataEC50:  1.65E+3nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457546(CHEMBL4206237)
Affinity DataEC50:  2nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor beta(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457547(CHEMBL3953756)
Affinity DataEC50:  40nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARbeta (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457561(CHEMBL3916016)
Affinity DataEC50:  200nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457551(CHEMBL4217953)
Affinity DataEC50:  34nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM31888(CD666)
Affinity DataEC50:  46nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457558(CHEMBL4203950)
Affinity DataEC50:  422nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457557(CHEMBL4215630)
Affinity DataEC50:  120nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457556(CHEMBL4217018)
Affinity DataEC50:  47nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457555(CHEMBL4214493)
Affinity DataEC50:  60nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457554(CHEMBL4202830)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457553(CHEMBL4210099)
Affinity DataEC50:  4.40nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Nestle Skin Health

Curated by ChEMBL
LigandPNGBDBM50457552(CHEMBL4210595)
Affinity DataEC50:  0.220nMAssay Description:Agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
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