Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50001201
TargetG-protein coupled bile acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM50271977(CHEMBL4127558)
Affinity DataEC50: >100nMAssay Description:Agonist activity at human TGR5 expressed in CHOK1 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM50271983(CHEMBL4128655)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human TGR5 expressed in CHOK1 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM50271984(CHEMBL4128688)
Affinity DataEC50:  68nMAssay Description:Agonist activity at human TGR5 expressed in CHOK1 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM50271985(CHEMBL4126485)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human TGR5 expressed in CHOK1 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM50271986(CHEMBL4129882)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human TGR5 expressed in CHOK1 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM50271987(CHEMBL4126607)
Affinity DataEC50: >100nMAssay Description:Agonist activity at human TGR5 expressed in CHOK1 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM50271995(CHEMBL4130025)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human TGR5 expressed in CHOK1 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM50271996(CHEMBL4130175)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human TGR5 expressed in CHOK1 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM50271997(CHEMBL4128816)
Affinity DataEC50:  95nMAssay Description:Agonist activity at human TGR5 expressed in CHOK1 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM50271998(CHEMBL4127302)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at human TGR5 expressed in CHOK1 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM50272007(CHEMBL4127444)
Affinity DataEC50:  36nMAssay Description:Agonist activity at human TGR5 expressed in CHOK1 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM50272009(CHEMBL4126062)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human TGR5 expressed in CHOK1 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM50161834(CHEMBL3794175)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human TGR5 expressed in CHOK1 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed