Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50002168
TargetPlatelet-activating factor acetylhydrolase(Human)
University of Reunion

Curated by ChEMBL
LigandPNGBDBM50125265(N-(2-Diethylamino-ethyl)-2-[2-(4-fluoro-benzylsulf...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Lp-PLA2 in human plasma LDL fractions using 2-thio platelet-activating factor as substrate by TMB dye based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
University of Reunion

Curated by ChEMBL
LigandPNGBDBM50125265(N-(2-Diethylamino-ethyl)-2-[2-(4-fluoro-benzylsulf...)
Affinity DataIC50: 0.25nMAssay Description:Inhibition of human Lp-PLA2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
University of Reunion

Curated by ChEMBL
LigandPNGBDBM50454544(CHEMBL4208988)
Affinity DataIC50: 52nMAssay Description:Inhibition of Lp-PLA2 in human plasma LDL fractions using 2-thio platelet-activating factor as substrate by TMB dye based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
University of Reunion

Curated by ChEMBL
LigandPNGBDBM50454545(CHEMBL4211451)
Affinity DataIC50: 100nMAssay Description:Inhibition of Lp-PLA2 in human plasma LDL fractions using 2-thio platelet-activating factor as substrate by TMB dye based spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed