Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50046385
LigandPNGBDBM50109198(CHEMBL3601091)
Affinity DataEC50:  1.98E+3nMAssay Description:Agonist activity at human PPARalpha transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109262(CHEMBL3601088)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109200(CHEMBL3601089)
Affinity DataEC50:  1.62E+3nMAssay Description:Agonist activity at human PPARgamma transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109199(CHEMBL3601090)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109196(CHEMBL3601092)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50099491(cid_3392731 | CHEMBL21241 | 2-(4-{2-[3-Cyclohexyl-...)
Affinity DataEC50:  6.5nMAssay Description:Agonist activity at human PPARalpha transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM29080(Oleamide MEA | Oleoyl monoethanolamide | CHEMBL280...)
Affinity DataEC50:  152nMAssay Description:Agonist activity at human PPARalpha transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109159(CHEMBL3600934)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARalpha transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109158(CHEMBL3601087)
Affinity DataEC50:  670nMAssay Description:Agonist activity at human PPARalpha transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109262(CHEMBL3601088)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARalpha transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109200(CHEMBL3601089)
Affinity DataEC50:  821nMAssay Description:Agonist activity at human PPARalpha transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109199(CHEMBL3601090)
Affinity DataEC50:  6.62E+3nMAssay Description:Agonist activity at human PPARalpha transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109158(CHEMBL3601087)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at human PPARgamma transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109196(CHEMBL3601092)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARalpha transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109166(CHEMBL3601093)
Affinity DataEC50:  756nMAssay Description:Agonist activity at human PPARalpha transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109165(CHEMBL3601094)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARalpha transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109164(CHEMBL3601095)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARalpha transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109163(CHEMBL3601096)
Affinity DataEC50:  966nMAssay Description:Agonist activity at human PPARalpha transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109162(CHEMBL3601097)
Affinity DataEC50:  1.92E+3nMAssay Description:Agonist activity at human PPARalpha transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109161(CHEMBL3601098)
Affinity DataEC50:  866nMAssay Description:Agonist activity at human PPARalpha transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50109160(CHEMBL3601099)
Affinity DataEC50:  981nMAssay Description:Agonist activity at human PPARalpha transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed
LigandPNGBDBM50030474(US9562012, rosiglitazone | CHEBI:50122 | Avandamet...)
Affinity DataEC50:  87nMAssay Description:Agonist activity at human PPARgamma transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50109159(CHEMBL3600934)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma transfected in human MCF7 cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2016
Entry Details Article
PubMed