Report error Found 112 Enz. Inhib. hit(s) with all data for entry = 50006159
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 4.90E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 310nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 990nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 3.30E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 1.30E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 3.80E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 1.30E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 660nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 270nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 890nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 460nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 520nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 780nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 780nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 730nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 3.80E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 2.90E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 270nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 310nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 4.90E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 1.80E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 890nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 2.30E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 910nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 2.90E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 3.90E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 2.30E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 2.00E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 1.90E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 850nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 1.50E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 2.80E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 6.30E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 150nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 2.20E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 3.60E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 1.90E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 1.80E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 4(Human)
Northwest A&F University
Curated by ChEMBL
Northwest A&F University
Curated by ChEMBL
Affinity DataEC50: 3.70E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair



























