Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50045209
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50050071(CHEMBL3317729)
Affinity DataIC50: 46nMAssay Description:Inhibition of mGluR5 in rat embryo neuronal culture assessed as calcium level by Fluo-4/AM dye based fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50050067(CHEMBL3317720)
Affinity DataIC50: 150nMAssay Description:Inhibition of mGluR5 in rat embryo neuronal culture assessed as calcium level by Fluo-4/AM dye based fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50050070(CHEMBL3317727)
Affinity DataIC50: 350nMAssay Description:Inhibition of mGluR5 in rat embryo neuronal culture assessed as calcium level by Fluo-4/AM dye based fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50050066(CHEMBL3317710)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mGluR5 in rat embryo neuronal culture assessed as calcium level by Fluo-4/AM dye based fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50049951(CHEMBL3317708)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of mGluR5 in rat embryo neuronal culture assessed as calcium level by Fluo-4/AM dye based fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50049953(CHEMBL3317706)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of mGluR5 in rat embryo neuronal culture assessed as calcium level by Fluo-4/AM dye based fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50049952(CHEMBL3317707)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of mGluR5 in rat embryo neuronal culture assessed as calcium level by Fluo-4/AM dye based fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50050071(CHEMBL3317729)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50050067(CHEMBL3317720)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50050070(CHEMBL3317727)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50050069(CHEMBL3317726)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50050066(CHEMBL3317710)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50050065(CHEMBL3317709)
Affinity DataKi:  224nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50050068(CHEMBL3317721)
Affinity DataKi:  311nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50049951(CHEMBL3317708)
Affinity DataKi:  343nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50049953(CHEMBL3317706)
Affinity DataKi:  730nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50049952(CHEMBL3317707)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [3H]-M-MPEP from mGluR5 in rat cerebrocortical membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed