Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50032978
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337290(S-5-Methoxy-9-(3-(4-(3-aminopropyl)piperazin-1-yl)...)
Affinity DataEC50:  466nMAssay Description:Agonist activity at human MC4 receptor expressed in BHK cells assessed as stimulation of agonist-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337289(N-[(13S)-15-{3-[4-(3-aminopropyl)piperazin-1-yl]pr...)
Affinity DataEC50:  697nMAssay Description:Agonist activity at human MC4 receptor expressed in BHK cells assessed as stimulation of agonist-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337290(S-5-Methoxy-9-(3-(4-(3-aminopropyl)piperazin-1-yl)...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human MC1 receptor expressed in BHK cells assessed as stimulation of agonist-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337289(N-[(13S)-15-{3-[4-(3-aminopropyl)piperazin-1-yl]pr...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human MC1 receptor expressed in BHK cells assessed as stimulation of agonist-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337290(S-5-Methoxy-9-(3-(4-(3-aminopropyl)piperazin-1-yl)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human MC3 receptor expressed in BHK cells assessed as stimulation of agonist-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337289(N-[(13S)-15-{3-[4-(3-aminopropyl)piperazin-1-yl]pr...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human MC3 receptor expressed in BHK cells assessed as stimulation of agonist-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337289(N-[(13S)-15-{3-[4-(3-aminopropyl)piperazin-1-yl]pr...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human MC5 receptor expressed in BHK cells assessed as stimulation of agonist-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337290(S-5-Methoxy-9-(3-(4-(3-aminopropyl)piperazin-1-yl)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human MC5 receptor expressed in BHK cells assessed as stimulation of agonist-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337290(S-5-Methoxy-9-(3-(4-(3-aminopropyl)piperazin-1-yl)...)
Affinity DataKi:  116nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337289(N-[(13S)-15-{3-[4-(3-aminopropyl)piperazin-1-yl]pr...)
Affinity DataKi:  328nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337290(S-5-Methoxy-9-(3-(4-(3-aminopropyl)piperazin-1-yl)...)
Affinity DataKi:  388nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337290(S-5-Methoxy-9-(3-(4-(3-aminopropyl)piperazin-1-yl)...)
Affinity DataKi:  392nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337289(N-[(13S)-15-{3-[4-(3-aminopropyl)piperazin-1-yl]pr...)
Affinity DataKi:  403nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337290(S-5-Methoxy-9-(3-(4-(3-aminopropyl)piperazin-1-yl)...)
Affinity DataKi:  1.18E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337289(N-[(13S)-15-{3-[4-(3-aminopropyl)piperazin-1-yl]pr...)
Affinity DataKi:  1.53E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337289(N-[(13S)-15-{3-[4-(3-aminopropyl)piperazin-1-yl]pr...)
Affinity DataKi:  4.53E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed