Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50028419
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249516(cis-2-(4-((3S,5S)-5-(3,3-difluoropyrrolidine-1-car...)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249548(cis-(3,3-difluoropyrrolidin-1-yl)((2S,4S)-4-(4-(ox...)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249515(cis-(3,3-difluoropyrrolidin-1-yl)((2S,4S)-4-(4-(5-...)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249514(cis-(3,3-difluoropyrrolidin-1-yl)((2S,4S)-4-(4-(py...)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249513(cis-(3,3-difluoropyrrolidin-1-yl)((2S,4S)-4-(4-(ox...)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249512(cis-(3,3-difluoropyrrolidin-1-yl)((2S,4S)-4-(4-(ox...)
Affinity DataIC50: 7.40nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249481(cis-((2S,4S)-4-(4-(benzo[d]oxazol-2-yl)piperazin-1...)
Affinity DataIC50: 8.20nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249480(cis-((2S,4S)-4-(4-(benzo[d]isoxazol-3-yl)piperazin...)
Affinity DataIC50: 8.70nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249479(PF-00734200 | cis-(3,3-Difluoro-pyrrolidin-1-yl)-[...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249479(PF-00734200 | cis-(3,3-Difluoro-pyrrolidin-1-yl)-[...)
Affinity DataIC50: 13nMAssay Description:Inhibition of rat plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249479(PF-00734200 | cis-(3,3-Difluoro-pyrrolidin-1-yl)-[...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249552(cis-((3S,4R)-3,4-difluoropyrrolidin-1-yl)((2S,4S)-...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249098(cis-((2S,4S)-4-(4-(pyrimidin-2-yl)piperazin-1-yl)p...)
Affinity DataIC50: 25nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249549(cis-((2S,4S)-4-(4-(pyrimidin-2-yl)piperazin-1-yl)p...)
Affinity DataIC50: 31nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249551(cis-((S)-3-fluoropyrrolidin-1-yl)((2S,4S)-4-(4-(py...)
Affinity DataIC50: 31nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249100(cis-(3-fluoroazetidin-1-yl)((2S,4S)-4-(4-(pyrimidi...)
Affinity DataIC50: 41nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249550(cis-((R)-3-fluoropyrrolidin-1-yl)((2S,4S)-4-(4-(py...)
Affinity DataIC50: 51nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249101(cis-(3,3-difluoroazetidin-1-yl)((2S,4S)-4-(4-(pyri...)
Affinity DataIC50: 134nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249516(cis-2-(4-((3S,5S)-5-(3,3-difluoropyrrolidine-1-car...)
Affinity DataIC50: 210nMAssay Description:Inhibition of human recombinant DPP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249099(cis-azetidin-1-yl((2S,4S)-4-(4-(pyrimidin-2-yl)pip...)
Affinity DataIC50: 309nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249097(cis-((3R,4R)-3,4-difluoropyrrolidin-1-yl)((2S,4S)-...)
Affinity DataIC50: 309nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249137(trans-(3,3-difluoropyrrolidin-1-yl)((2S,4R)-4-(4-(...)
Affinity DataIC50: 338nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249515(cis-(3,3-difluoropyrrolidin-1-yl)((2S,4S)-4-(4-(5-...)
Affinity DataIC50: 530nMAssay Description:Inhibition of human recombinant DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249514(cis-(3,3-difluoropyrrolidin-1-yl)((2S,4S)-4-(4-(py...)
Affinity DataIC50: 540nMAssay Description:Inhibition of human recombinant DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249514(cis-(3,3-difluoropyrrolidin-1-yl)((2S,4S)-4-(4-(py...)
Affinity DataIC50: 660nMAssay Description:Inhibition of human recombinant DPP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249515(cis-(3,3-difluoropyrrolidin-1-yl)((2S,4S)-4-(4-(5-...)
Affinity DataIC50: 660nMAssay Description:Inhibition of human recombinant DPP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249512(cis-(3,3-difluoropyrrolidin-1-yl)((2S,4S)-4-(4-(ox...)
Affinity DataIC50: 970nMAssay Description:Inhibition of human recombinant DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249513(cis-(3,3-difluoropyrrolidin-1-yl)((2S,4S)-4-(4-(ox...)
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of human recombinant DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249480(cis-((2S,4S)-4-(4-(benzo[d]isoxazol-3-yl)piperazin...)
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of human recombinant DPP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249480(cis-((2S,4S)-4-(4-(benzo[d]isoxazol-3-yl)piperazin...)
Affinity DataIC50: 2.24E+3nMAssay Description:Inhibition of human recombinant DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249481(cis-((2S,4S)-4-(4-(benzo[d]oxazol-2-yl)piperazin-1...)
Affinity DataIC50: 2.26E+3nMAssay Description:Inhibition of human recombinant DPP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249548(cis-(3,3-difluoropyrrolidin-1-yl)((2S,4S)-4-(4-(ox...)
Affinity DataIC50: 2.39E+3nMAssay Description:Inhibition of human recombinant DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249098(cis-((2S,4S)-4-(4-(pyrimidin-2-yl)piperazin-1-yl)p...)
Affinity DataIC50: 2.46E+3nMAssay Description:Inhibition of human recombinant DPP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249481(cis-((2S,4S)-4-(4-(benzo[d]oxazol-2-yl)piperazin-1...)
Affinity DataIC50: 2.66E+3nMAssay Description:Inhibition of human recombinant DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249548(cis-(3,3-difluoropyrrolidin-1-yl)((2S,4S)-4-(4-(ox...)
Affinity DataIC50: 2.88E+3nMAssay Description:Inhibition of human recombinant DPP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249479(PF-00734200 | cis-(3,3-Difluoro-pyrrolidin-1-yl)-[...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human recombinant DPP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249479(PF-00734200 | cis-(3,3-Difluoro-pyrrolidin-1-yl)-[...)
Affinity DataIC50: 5.98E+3nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249479(PF-00734200 | cis-(3,3-Difluoro-pyrrolidin-1-yl)-[...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human recombinant DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249512(cis-(3,3-difluoropyrrolidin-1-yl)((2S,4S)-4-(4-(ox...)
Affinity DataIC50: 7.12E+3nMAssay Description:Inhibition of human recombinant DPP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249098(cis-((2S,4S)-4-(4-(pyrimidin-2-yl)piperazin-1-yl)p...)
Affinity DataIC50: 7.88E+3nMAssay Description:Inhibition of human recombinant DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249513(cis-(3,3-difluoropyrrolidin-1-yl)((2S,4S)-4-(4-(ox...)
Affinity DataIC50: 8.47E+3nMAssay Description:Inhibition of human recombinant DPP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249516(cis-2-(4-((3S,5S)-5-(3,3-difluoropyrrolidine-1-car...)
Affinity DataIC50: 9.15E+3nMAssay Description:Inhibition of human recombinant DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249549(cis-((2S,4S)-4-(4-(pyrimidin-2-yl)piperazin-1-yl)p...)
Affinity DataIC50: 9.69E+3nMAssay Description:Inhibition of human recombinant DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50249516(cis-2-(4-((3S,5S)-5-(3,3-difluoropyrrolidine-1-car...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG by patch-clamp techniqueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249550(cis-((R)-3-fluoropyrrolidin-1-yl)((2S,4S)-4-(4-(py...)
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of human recombinant DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249479(PF-00734200 | cis-(3,3-Difluoro-pyrrolidin-1-yl)-[...)
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of human FAP expressed in african green monkey COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249552(cis-((3S,4R)-3,4-difluoropyrrolidin-1-yl)((2S,4S)-...)
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of human recombinant DPP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249551(cis-((S)-3-fluoropyrrolidin-1-yl)((2S,4S)-4-(4-(py...)
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of human recombinant DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249552(cis-((3S,4R)-3,4-difluoropyrrolidin-1-yl)((2S,4S)-...)
Affinity DataIC50: 1.71E+4nMAssay Description:Inhibition of human recombinant DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249549(cis-((2S,4S)-4-(4-(pyrimidin-2-yl)piperazin-1-yl)p...)
Affinity DataIC50: 2.04E+4nMAssay Description:Inhibition of human recombinant DPP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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