Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50027011
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50265301(5-(4-phenoxybenzylidene)pyrimidine-2,4,6(1H,3H,5H)...)
Affinity DataIC50: 100nMAssay Description:Displacement of [3H]rosiglitazone from mouse PPARgamma receptor by scintillation proximation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50265171(4-(4-((2,4,6-trioxotetrahydropyrimidin-5(6H)-ylide...)
Affinity DataIC50: 200nMAssay Description:Displacement of [3H]rosiglitazone from mouse PPARgamma receptor by scintillation proximation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50265213(5-(4-((4-methoxyphenoxy)methyl)benzylidene)pyrimid...)
Affinity DataIC50: 200nMAssay Description:Displacement of [3H]rosiglitazone from mouse PPARgamma receptor by scintillation proximation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50265270(5-(4-((10H-phenoxazin-10-yl)methyl)benzylidene)pyr...)
Affinity DataIC50: 500nMAssay Description:Displacement of [3H]rosiglitazone from mouse PPARgamma receptor by scintillation proximation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50049240((+-)-5-((4-(2-(5-ethyl-2-pyridinyl)ethoxy)phenyl)m...)
Affinity DataIC50: 700nMAssay Description:Displacement of [3H]rosiglitazone from mouse PPARgamma receptor by scintillation proximation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50265211(5-(3-(2-(p-tolyloxy)ethoxy)benzylidene)pyrimidine-...)
Affinity DataIC50: 800nMAssay Description:Displacement of [3H]rosiglitazone from mouse PPARgamma receptor by scintillation proximation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50265212(5-(4-((4-nitrophenoxy)methyl)benzylidene)pyrimidin...)
Affinity DataIC50: 2.50E+3nMAssay Description:Displacement of [3H]rosiglitazone from mouse PPARgamma receptor by scintillation proximation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed