Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50025696
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataIC50: 1.90nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251131(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-N-cycloh...)
Affinity DataIC50: 49.4nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251130(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-Ncyclohe...)
Affinity DataIC50: 62.8nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242549(4-((2-Chlorophenyl)(4-chlorophenyl)methyl)-N-cyclo...)
Affinity DataIC50: 66.5nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242548(4-((2-Chlorophenyl)(4-chlorophenyl)methyl)-N-cyclo...)
Affinity DataIC50: 72.8nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251131(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-N-cycloh...)
Affinity DataIC50: 82.3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242557(4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-c...)
Affinity DataIC50: 89.2nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251130(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-Ncyclohe...)
Affinity DataIC50: 103nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242582(4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-c...)
Affinity DataIC50: 104nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242566(N-tert-Butyl-4-((2-chlorophenyl)(4-chlorophenyl)-m...)
Affinity DataIC50: 122nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251132(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-N-(cyclo...)
Affinity DataIC50: 127nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242548(4-((2-Chlorophenyl)(4-chlorophenyl)methyl)-N-cyclo...)
Affinity DataIC50: 128nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242601(4-((4-Chlorophenyl)(2-(trifluoromethyl)phenyl)-met...)
Affinity DataIC50: 141nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251132(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-N-(cyclo...)
Affinity DataIC50: 146nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242568(4-((4-Chlorophenyl)(o-tolyl)methyl)-N-cycloheptylp...)
Affinity DataIC50: 151nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242537(4-((4-Chlorophenyl)(2,3-dichlorophenyl)methyl)-N-c...)
Affinity DataIC50: 158nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242600(4-((4-Chlorophenyl)(2-(trifluoromethyl)phenyl)-met...)
Affinity DataIC50: 163nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242568(4-((4-Chlorophenyl)(o-tolyl)methyl)-N-cycloheptylp...)
Affinity DataIC50: 163nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242600(4-((4-Chlorophenyl)(2-(trifluoromethyl)phenyl)-met...)
Affinity DataIC50: 186nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242556(4-((4-Chlorophenyl)(2,3-dichlorophenyl)methyl)-N-c...)
Affinity DataIC50: 186nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242565(4-((2-Chlorophenyl)(4-chlorophenyl)methyl)-N-(cycl...)
Affinity DataIC50: 189nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242567(4-((4-Chlorophenyl)(o-tolyl)methyl)-N-cyclohexylpi...)
Affinity DataIC50: 195nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242601(4-((4-Chlorophenyl)(2-(trifluoromethyl)phenyl)-met...)
Affinity DataIC50: 204nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251117(2-(4-((2-Chlorophenyl)(4-chlorophenyl)methyl)-pipe...)
Affinity DataIC50: 226nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242549(4-((2-Chlorophenyl)(4-chlorophenyl)methyl)-N-cyclo...)
Affinity DataIC50: 226nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251118(2-(4-((2-Chlorophenyl)(4-chlorophenyl)methyl)-pipe...)
Affinity DataIC50: 229nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251133(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-N-tert-b...)
Affinity DataIC50: 237nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242567(4-((4-Chlorophenyl)(o-tolyl)methyl)-N-cyclohexylpi...)
Affinity DataIC50: 248nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242547(1-(4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-...)
Affinity DataIC50: 257nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242558(4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-(...)
Affinity DataIC50: 262nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242565(4-((2-Chlorophenyl)(4-chlorophenyl)methyl)-N-(cycl...)
Affinity DataIC50: 273nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251133(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-N-tert-b...)
Affinity DataIC50: 286nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242598(4-((4-Chlorophenyl)(o-tolyl)methyl)-N-(cyclohexylm...)
Affinity DataIC50: 291nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242539(N-tert-Butyl-4-((4-chlorophenyl)(2,3-dichloropheny...)
Affinity DataIC50: 316nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242599(N-tert-Butyl-4-((4-chlorophenyl)(o-tolyl)methyl)pi...)
Affinity DataIC50: 334nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242598(4-((4-Chlorophenyl)(o-tolyl)methyl)-N-(cyclohexylm...)
Affinity DataIC50: 340nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242582(4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-c...)
Affinity DataIC50: 367nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242537(4-((4-Chlorophenyl)(2,3-dichlorophenyl)methyl)-N-c...)
Affinity DataIC50: 424nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242556(4-((4-Chlorophenyl)(2,3-dichlorophenyl)methyl)-N-c...)
Affinity DataIC50: 441nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242566(N-tert-Butyl-4-((2-chlorophenyl)(4-chlorophenyl)-m...)
Affinity DataIC50: 443nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251115(4-((4-Chlorophenyl)(2-(trifluoromethyl)phenyl)-met...)
Affinity DataIC50: 526nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242599(N-tert-Butyl-4-((4-chlorophenyl)(o-tolyl)methyl)pi...)
Affinity DataIC50: 680nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242557(4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-c...)
Affinity DataIC50: 729nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242539(N-tert-Butyl-4-((4-chlorophenyl)(2,3-dichloropheny...)
Affinity DataIC50: 783nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251115(4-((4-Chlorophenyl)(2-(trifluoromethyl)phenyl)-met...)
Affinity DataIC50: 798nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242581(4-(Bis(4-chlorophenyl)methyl)-N-cyclohexylpiperazi...)
Affinity DataIC50: 914nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242558(4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-(...)
Affinity DataIC50: 1.04E+3nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242584((4-(Bis(4-chlorophenyl)methyl)piperazin-1-yl)-(cyc...)
Affinity DataIC50: 1.07E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50242585(1-(4-(Bis(4-chlorophenyl)methyl)piperazin-1-yl)-he...)
Affinity DataIC50: 1.15E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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