Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50020260
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211814(4-(2-(4-fluorophenyl)-7-((isopropylamino)methyl)H-...)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211811(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211805(4-(7-(((3-(dimethylamino)propyl)(methyl)amino)meth...)
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50182359(N-benzyl-4-(7-((dimethylamino)methyl)-2-(4-fluorop...)
Affinity DataIC50: 0.0810nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211820(4-(7-(((2-(azetidin-1-yl)ethyl)(methyl)amino)methy...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211802(2-(((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethylami...)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211812(4-(2-(4-fluorophenyl)-7-((isopropyl(methyl)amino)m...)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211803(4-(7-((ethyl(methyl)amino)methyl)-2-(4-fluoropheny...)
Affinity DataIC50: 0.130nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211808(N-(2-(((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethyl...)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211821(2-(((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethylami...)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211819(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211816((S)-2-(((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethy...)
Affinity DataIC50: 0.260nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211810(4-(2-(4-fluorophenyl)-7-((methyl((tetrahydrofuran-...)
Affinity DataIC50: 0.270nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50182361(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50: 0.280nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211823(4-(7-((ethyl(methyl)amino)methyl)-2-(4-fluoropheny...)
Affinity DataIC50: 0.290nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211818(N-tert-butyl-4-(7-((dimethylamino)methyl)-2-(4-flu...)
Affinity DataIC50: 0.310nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211822(2-(((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethylami...)
Affinity DataIC50: 0.390nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211817(4-(7-(azetidin-1-ylmethyl)-2-(4-fluorophenyl)H-imi...)
Affinity DataIC50: 0.450nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211815(1-(azetidin-1-yl)-2-(((2-(4-fluorophenyl)-3-(2-((S...)
Affinity DataIC50: 0.570nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211806(4-(2-(4-fluorophenyl)-7-((isopropyl(methyl)amino)m...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211809(4-(7-(azetidin-1-ylmethyl)-2-(4-fluorophenyl)H-imi...)
Affinity DataIC50: 0.860nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211807(4-(2-(4-fluorophenyl)-7-((isopropyl(methyl)amino)m...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211813(N-tert-butyl-4-(2-(4-fluorophenyl)-7-((isopropyl(m...)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211804(ethyl 4-((2-(4-fluorophenyl)-3-(2-((S)-1-phenyleth...)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed