Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50016042
TargetCoagulation factor XIII A chain(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164227(5-Methyl-2-(2-oxo-propylsulfanyl)-thiazolo[2,3-b][...)
Affinity DataIC50: 100nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164216(N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-methyl-...)
Affinity DataIC50: 110nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164222(N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-ylamino)-h...)
Affinity DataIC50: 130nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164227(5-Methyl-2-(2-oxo-propylsulfanyl)-thiazolo[2,3-b][...)
Affinity DataIC50: 250nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164223(2-{Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-[6-(2-nitr...)
Affinity DataIC50: 420nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164224({Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-[6-(2-nitro-...)
Affinity DataIC50: 620nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164225(N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-ylamino)-h...)
Affinity DataIC50: 700nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164226(N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-ylamino)-h...)
Affinity DataIC50: 910nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164218(N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-ylamino)-h...)
Affinity DataIC50: 1.90E+3nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164221(N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-ylamino)-h...)
Affinity DataIC50: 2.20E+3nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164219(N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-ylamino)-h...)
Affinity DataIC50: 2.30E+3nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164216(N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-methyl-...)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164222(N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-ylamino)-h...)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164217(N*1*-Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-hexane-1...)
Affinity DataIC50: 1.10E+4nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164224({Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-[6-(2-nitro-...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164223(2-{Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-[6-(2-nitr...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibitory concentration against guinea pig liver transglutaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164220(N-Hexyl-2-nitro-benzenesulfonamide | CHEMBL192376)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor XIII A chain(Human)
Apotex Research

Curated by ChEMBL
LigandPNGBDBM50164215(2-Nitro-N-[6-(3-nitro-pyridin-2-ylamino)-hexyl]-be...)
Affinity DataIC50: 1.70E+5nMAssay Description:In vitro inhibitory concentration of compound against factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed