Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50010682
Target72 kDa type IV collagenase(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50097588((R)-(4-Hydroxy-cyclohexyl)-(4'-methoxy-biphenyl-4-...)
Affinity DataIC50: 12nMAssay Description:Inhibition of gelatinase A (Matrix metalloprotease-2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50097589((R)-((S)-4-Hydroxy-cyclohex-2-enyl)-(4'-methoxy-bi...)
Affinity DataIC50: 20nMAssay Description:Inhibition of gelatinase A (Matrix metalloprotease-2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50097588((R)-(4-Hydroxy-cyclohexyl)-(4'-methoxy-biphenyl-4-...)
Affinity DataIC50: 30nMAssay Description:Inhibition of Collagenase 3 (Matrix metalloprotease-13)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50097587((R)-((S)-2-Bromo-4-hydroxy-cyclohex-2-enyl)-(4'-me...)
Affinity DataIC50: 38nMAssay Description:Inhibition of gelatinase A (Matrix metalloprotease-2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50097587((R)-((S)-2-Bromo-4-hydroxy-cyclohex-2-enyl)-(4'-me...)
Affinity DataIC50: 131nMAssay Description:Inhibition of Collagenase 3 (Matrix metalloprotease-13)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50097589((R)-((S)-4-Hydroxy-cyclohex-2-enyl)-(4'-methoxy-bi...)
Affinity DataIC50: 176nMAssay Description:Inhibition of Collagenase 3 (Matrix metalloprotease-13)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50097590(2-(4-Hydroxy-cyclohexyl)-2-(4'-methoxy-biphenyl-4-...)
Affinity DataIC50: 251nMAssay Description:Inhibition of gelatinase A (Matrix metalloprotease-2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50097590(2-(4-Hydroxy-cyclohexyl)-2-(4'-methoxy-biphenyl-4-...)
Affinity DataIC50: 338nMAssay Description:Inhibition of Collagenase 3 (Matrix metalloprotease-13)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50097588((R)-(4-Hydroxy-cyclohexyl)-(4'-methoxy-biphenyl-4-...)
Affinity DataIC50: 1.22E+3nMAssay Description:Inhibition of Stromelysin (Matrix metalloprotease-3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50097589((R)-((S)-4-Hydroxy-cyclohex-2-enyl)-(4'-methoxy-bi...)
Affinity DataIC50: 2.49E+3nMAssay Description:Inhibition of Stromelysin (Matrix metalloprotease-3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50097587((R)-((S)-2-Bromo-4-hydroxy-cyclohex-2-enyl)-(4'-me...)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of Stromelysin (Matrix metalloprotease-3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50097590(2-(4-Hydroxy-cyclohexyl)-2-(4'-methoxy-biphenyl-4-...)
Affinity DataIC50: 6.15E+3nMAssay Description:Inhibition of Stromelysin (Matrix metalloprotease-3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed