Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50010641
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097007(4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 50nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096979(4-{4-[2-(2-Naphthalen-1-yl-1H-indol-3-yl)-ethylami...)
Affinity DataIC50: 130nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096995(4-(4-{2-[2-(3,5-Dichloro-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 170nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096982(4-{4-[2-(2-m-Tolyl-1H-indol-3-yl)-ethylamino]-buty...)
Affinity DataIC50: 200nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097011(4-(2-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 200nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096988(4-(5-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 200nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096998(4-(3-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 250nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097004(4-{4-[2-(2-Benzo[b]thiophen-3-yl-1H-indol-3-yl)-et...)
Affinity DataIC50: 300nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097017(4-(4-{2-[2-(2,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 400nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096978(4-{4-[2-(2-o-Tolyl-1H-indol-3-yl)-ethylamino]-buty...)
Affinity DataIC50: 500nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097013(4-(6-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 600nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096993(4-(4-{2-[2-(3-Methoxy-phenyl)-1H-indol-3-yl]-ethyl...)
Affinity DataIC50: 600nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097008(4-(4-{2-[2-(3,5-Dimethoxy-phenyl)-1H-indol-3-yl]-e...)
Affinity DataIC50: 700nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096989(4-(4-{2-[2-(2,3-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 900nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097012(4-(4-{2-[2-(3-Ethyl-phenyl)-1H-indol-3-yl]-ethylam...)
Affinity DataIC50: 900nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096990(4-{4-[2-(2-Phenyl-1H-indol-3-yl)-ethylamino]-butyl...)
Affinity DataIC50: 1.30E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096983(4-(4-{2-[2-(3,5-Bis-trifluoromethyl-phenyl)-1H-ind...)
Affinity DataIC50: 1.50E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096980(4-(4-{2-[2-(2,6-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 1.70E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096985(4-{4-[2-(2-Isoquinolin-5-yl-1H-indol-3-yl)-ethylam...)
Affinity DataIC50: 1.90E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096997(4-(4-{2-[2-(3,4-Dimethoxy-phenyl)-1H-indol-3-yl]-e...)
Affinity DataIC50: 2.00E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097000(4-(5-{2-[2-(3,4-Dimethoxy-phenyl)-1H-indol-3-yl]-e...)
Affinity DataIC50: 2.00E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097006(4-((R)-4-{2-[2-(3,4-Dimethoxy-phenyl)-1H-indol-3-y...)
Affinity DataIC50: 2.00E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096996(4-{4-[2-(2-Benzo[b]thiophen-2-yl-1H-indol-3-yl)-et...)
Affinity DataIC50: 2.50E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097010(4-{4-[2-(2-Naphthalen-2-yl-1H-indol-3-yl)-ethylami...)
Affinity DataIC50: 2.50E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096986(4-{4-[2-(1'-Methyl-1H,1'H-[2,5']biindolyl-3-yl)-et...)
Affinity DataIC50: 2.80E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096994(4-((R)-3-{2-[2-(3,4-Dimethoxy-phenyl)-1H-indol-3-y...)
Affinity DataIC50: 3.00E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097001(4-((S)-3-{2-[2-(3,4-Dimethoxy-phenyl)-1H-indol-3-y...)
Affinity DataIC50: 3.00E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097014(4-(2-{2-[2-(3,4-Dimethoxy-phenyl)-1H-indol-3-yl]-e...)
Affinity DataIC50: 4.00E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096991({2-[2-(3,4-Dimethoxy-phenyl)-1H-indol-3-yl]-ethyl}...)
Affinity DataIC50: 5.00E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096981(4-(3-{2-[2-(3,4-Dimethoxy-phenyl)-1H-indol-3-yl]-e...)
Affinity DataIC50: 6.00E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097003(4-({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethy...)
Affinity DataIC50: 9.00E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096992(4-{4-[2-(2-p-Tolyl-1H-indol-3-yl)-ethylamino]-buty...)
Affinity DataIC50: 9.00E+3nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097002(4-(6-{2-[2-(3,4-Dimethoxy-phenyl)-1H-indol-3-yl]-e...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097015(4-(4-{2-[2-(3,4-Dimethoxy-phenyl)-1H-indol-3-yl]-e...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096999(4-(4-{2-[2-(4-Fluoro-phenyl)-1H-indol-3-yl]-ethyla...)
Affinity DataIC50: 1.10E+4nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097016(4-({2-[2-(3,4-Dimethoxy-phenyl)-1H-indol-3-yl]-eth...)
Affinity DataIC50: 2.00E+4nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097009(4-(4-Amino-phenyl)-N-{2-[2-(3,4-dimethoxy-phenyl)-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096987(N-{2-[2-(3,4-Dimethoxy-phenyl)-1H-indol-3-yl]-ethy...)
Affinity DataIC50: 3.00E+4nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50096984(N-{2-[2-(3,4-Dimethoxy-phenyl)-1H-indol-3-yl]-ethy...)
Affinity DataIC50: 3.00E+4nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097005([4-(4-Benzyloxy-phenyl)-butyl]-{2-[2-(3,4-dimethox...)
Affinity DataIC50: 3.00E+4nMAssay Description:Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed