Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50009944
TargetB1 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089314(H-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-OH(JMV1645) | C...)
Affinity DataKi:  0.0230nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089307(H-Lys-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-OH(JMV1639)...)
Affinity DataKi:  0.0350nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089308(H-DArg-Arg-Pro-Hyp-Gly-Thi-Ser-DTic-Oic-Arg-OH( HO...)
Affinity DataKi:  0.0800nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50049949(2-(2-{[1-(2-{2-[2-({1-[1-(2-Amino-5-guanidino-pent...)
Affinity DataKi:  0.110nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089313(H-Lys-Arg-Pro-Hyp-Gly-Thi-Ser-D-BT-OH(JMV1669) | C...)
Affinity DataKi:  0.220nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089313(H-Lys-Arg-Pro-Hyp-Gly-Thi-Ser-D-BT-OH(JMV1669) | C...)
Affinity DataKi:  0.400nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089310(2-({1-[2-(2-{2-[(1-{1-[2-(2,6-Diamino-hexanoylamin...)
Affinity DataKi:  0.900nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089312(H-DArg-Arg-Pro-Hyp-Gly-Thi-Ser-D-BT-OH(JMV1431) | ...)
Affinity DataKi:  4.40nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089309(H-DArg-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-OH(JMV1638) | ...)
Affinity DataKi:  5.60nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089314(H-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-OH(JMV1645) | C...)
Affinity DataKi:  9.20nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089310(2-({1-[2-(2-{2-[(1-{1-[2-(2,6-Diamino-hexanoylamin...)
Affinity DataKi: >10nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089308(H-DArg-Arg-Pro-Hyp-Gly-Thi-Ser-DTic-Oic-Arg-OH( HO...)
Affinity DataKi: >10nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50049949(2-(2-{[1-(2-{2-[2-({1-[1-(2-Amino-5-guanidino-pent...)
Affinity DataKi: >10nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089306(2-{[1-(2-{2-[2-({1-[1-(2-Amino-5-guanidino-pentano...)
Affinity DataKi: >10nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089311(H-DArg-Arg-Pro-Hyp-Gly-Thi-Ser-D-Tic-Oic-OH ([des-...)
Affinity DataKi:  24nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089307(H-Lys-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-OH(JMV1639)...)
Affinity DataKi:  62nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089312(H-DArg-Arg-Pro-Hyp-Gly-Thi-Ser-D-BT-OH(JMV1431) | ...)
Affinity DataKi:  83nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089309(H-DArg-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-OH(JMV1638) | ...)
Affinity DataKi:  325nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089306(2-{[1-(2-{2-[2-({1-[1-(2-Amino-5-guanidino-pentano...)
Affinity DataKi:  382nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed