Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50009092
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.440nMAssay Description:Displacement of [3H]raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM55121(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080053(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080047((4-Methoxy-benzyl)-((R)-5-methoxy-1,2,3,4-tetrahyd...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50053670(CHEMBL541858 | CHEMBL69985 | ((R)-5-Fluoro-1,2,3,4...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080048((4-Fluoro-benzyl)-((R)-5-methoxy-1,2,3,4-tetrahydr...)
Affinity DataKi:  43.8nMAssay Description:Displacement of [3H]raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080053(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080050(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080047((4-Methoxy-benzyl)-((R)-5-methoxy-1,2,3,4-tetrahyd...)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080051(Benzyl-((R)-5-methoxy-1,2,3,4-tetrahydro-naphthale...)
Affinity DataKi:  65.6nMAssay Description:Displacement of [3H]raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080048((4-Fluoro-benzyl)-((R)-5-methoxy-1,2,3,4-tetrahydr...)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080051(Benzyl-((R)-5-methoxy-1,2,3,4-tetrahydro-naphthale...)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080055(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  82.3nMAssay Description:Displacement of [3H]quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080055(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  114nMAssay Description:Displacement of [3H]raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080052(Furan-2-ylmethyl-((R)-5-methoxy-1,2,3,4-tetrahydro...)
Affinity DataKi:  118nMAssay Description:Displacement of [3H]quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080052(Furan-2-ylmethyl-((R)-5-methoxy-1,2,3,4-tetrahydro...)
Affinity DataKi:  125nMAssay Description:Displacement of [3H]raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080049(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  152nMAssay Description:Displacement of [3H]raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054337(Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataKi:  179nMAssay Description:Inhibition of [3H]quinpirole binding to human dopamine D2A receptor expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50053670(CHEMBL541858 | CHEMBL69985 | ((R)-5-Fluoro-1,2,3,4...)
Affinity DataKi:  201nMAssay Description:Displacement of [3H]raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080050(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  215nMAssay Description:Displacement of [3H]quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080049(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  339nMAssay Description:Displacement of [3H]quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054337(Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataKi:  415nMAssay Description:Inhibition of [3H]raclopride binding to human dopamine D2A receptor expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM55121(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Affinity DataKi:  759nMAssay Description:Displacement of [3H]raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080056(Benzyl-((R)-5-methoxy-1,2,3,4-tetrahydro-naphthale...)
Affinity DataKi:  1.01E+3nMAssay Description:Displacement of [3H]raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080056(Benzyl-((R)-5-methoxy-1,2,3,4-tetrahydro-naphthale...)
Affinity DataKi:  1.31E+3nMAssay Description:Displacement of [3H]quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080054(Dibenzyl-((R)-5-methoxy-1,2,3,4-tetrahydro-naphtha...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080054(Dibenzyl-((R)-5-methoxy-1,2,3,4-tetrahydro-naphtha...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed