Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50008930
TargetVasopressin V2 receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50078646(N-[4-(4,10-Dihydro-1-thia-9-aza-benzo[f]azulene-9-...)
Affinity DataIC50: 0.700nMAssay Description:In vitro inhibition of [3H]AVP binding to human V2 receptor from murine fibroblast cell line (LV2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50065115(N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 1.20nMAssay Description:In vitro inhibition of [3H]AVP binding to human V2 receptor from murine fibroblast cell line (LV2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50078649(N-[3-Chloro-4-(4,10-dihydro-1-thia-9-aza-benzo[f]a...)
Affinity DataIC50: 6.80nMAssay Description:In vitro inhibition of [3H]AVP binding to human V2 receptor from murine fibroblast cell line (LV2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50078646(N-[4-(4,10-Dihydro-1-thia-9-aza-benzo[f]azulene-9-...)
Affinity DataIC50: 8.5nMAssay Description:In vitro inhibition of [3H]- AVP binding to V1a receptor from human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50078647(N-[4-(4,10-Dihydro-3-thia-9-aza-benzo[f]azulene-9-...)
Affinity DataIC50: 9nMAssay Description:In vitro inhibition of [3H]AVP binding to human V2 receptor from murine fibroblast cell line (LV2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50078648(2,4-Dichloro-N-[4-(4,10-dihydro-1-thia-9-aza-benzo...)
Affinity DataIC50: 19nMAssay Description:In vitro inhibition of [3H]AVP binding to human V2 receptor from murine fibroblast cell line (LV2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50078645(N-[5-(4,10-Dihydro-1-thia-9-aza-benzo[f]azulene-9-...)
Affinity DataIC50: 29nMAssay Description:In vitro inhibition of [3H]AVP binding to rat V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50078647(N-[4-(4,10-Dihydro-3-thia-9-aza-benzo[f]azulene-9-...)
Affinity DataIC50: 36nMAssay Description:In vitro inhibition of [3H]- AVP binding to V1a receptor from human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50078648(2,4-Dichloro-N-[4-(4,10-dihydro-1-thia-9-aza-benzo...)
Affinity DataIC50: 43nMAssay Description:In vitro inhibition of [3H]- AVP binding to V1a receptor from human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50078645(N-[5-(4,10-Dihydro-1-thia-9-aza-benzo[f]azulene-9-...)
Affinity DataIC50: 59nMAssay Description:In vitro inhibition of [3H]- AVP binding to rat V1a receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50065115(N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 230nMAssay Description:In vitro inhibition of [3H]- AVP binding to V1a receptor from human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed