BDBM481683 N1-cyclopentyl-N4,N4-bis(4- fluorobenzyl)benzene-1,4- disulfonamide::US10913710, Compound 93

SMILES Fc1ccc(CN(Cc2ccc(F)cc2)S(=O)(=O)c2ccc(cc2)S(=O)(=O)NC2CCCC2)cc1

InChI Key InChIKey=JTGWDAJVYKWFFD-UHFFFAOYSA-N

Data  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 481683   

TargetRetinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta(Human)
Max-Planck-Gesellschaft Zur Forderung Der Wissenschaften

US Patent
LigandPNGBDBM481683(N1-cyclopentyl-N4,N4-bis(4- fluorobenzyl)benzene-1...)
Affinity DataKd:  550nMAssay Description:Binding to PDEδ was validated and quantified by means of a displacement assay employing a fluorescent-tagged analog of the HMG-CoA reductase inh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2021
Entry Details
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