BDBM27277 indole derivative, 1c::tert-butyl 2-(2-benzenesulfonamido-2,3-dihydro-1H-inden-5-yl)-5-hydroxy-1H-indole-1-carboxylate

SMILES CC(C)(C)OC(=O)n1c(cc2cc(O)ccc12)-c1ccc2CC(Cc2c1)NS(=O)(=O)c1ccccc1

InChI Key InChIKey=GPMOKHWGTGSTLL-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 27277   

TargetOxysterols receptor LXR-beta(Human)
Tanabe Research Laboratories Usa

LigandPNGBDBM27277(tert-butyl 2-(2-benzenesulfonamido-2,3-dihydro-1H-...)
Affinity DataEC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2009
Entry Details Article
PubMed